SCHEMBL7408043

SCHEMBL7408043

COc1cc2c(cc1C(F)(F)F)N(C(=O)Nc1ccc(Oc3cccnc3)nc1)CC2.Nc1ccc(Oc2cccnc2)nc1

nearest known ligand 0.91

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 20/20 0.91
HTR2A P28223 17/20 0.91
HTR2B P41595 15/20 0.91
CYP1A2 P05177 9/20 0.91
CYP2C9 P11712 3/20 0.63
HTR6 P50406 1/20 0.63
CYP2D6 P10635 2/20 0.61
KDM4E B2RXH2 1/20 0.61
MEN1 O00255 1/20 0.61
GMNN O75496 1/20 0.61
LMNA P02545 1/20 0.61
TP53 P04637 1/20 0.61
CYP3A4 P08684 1/20 0.61
MAPT P10636 1/20 0.61
ALOX15 P16050 1/20 0.61
TSHR P16473 1/20 0.61
NFKB1 P19838 1/20 0.61
CYP2C19 P33261 1/20 0.61
THPO P40225 1/20 0.61
BLM P54132 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7082946 0.95 HTR2C (1.00) HTR2CHTR2AHTR2BCYP1A2CYP2C9
SCHEMBL7112081 0.86 HTR2C (0.82) HTR2CHTR2AHTR2BCYP1A2CYP2C9
SCHEMBL7379147 0.85 HTR2C (0.66) HTR2CHTR2AHTR2BCYP1A2
SCHEMBL7105805 0.85 HTR2C (0.80) HTR2CHTR2AHTR2BCYP1A2CYP2C9
SCHEMBL7078894 0.84 HTR2C (1.00) HTR2CHTR2AHTR2BCYP1A2CYP2C9
SCHEMBL7084100 0.84 HTR2C (0.78) HTR2CHTR2AHTR2BCYP1A2CYP2C9
SCHEMBL7039444 0.83 HTR2C (1.00) HTR2CHTR2AHTR2BCYP1A2CYP2C9
SCHEMBL7379418 0.80 HTR2C (0.91) HTR2CHTR2AHTR2BCYP1A2CYP2C9
SCHEMBL7082693 0.80 HTR2C (0.75) HTR2CHTR2AHTR2BCYP1A2CYP2C9
SCHEMBL7082972 0.80 HTR2C (0.72) HTR2CHTR2AHTR2BCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996023783-A1 INDOLE DERIVATIVES AS 5-HT RECEPTOR ANTAGONIST SMITHKLINE BEECHAM PLC (GB) 1996-08-08 WO disclosed