SCHEMBL740934

SCHEMBL740934

CCC(=O)Nc1ccc(NC(=O)COc2ccc(C)cc2C)cc1

nearest known ligand 0.74

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.70
ALDH1A1 P00352 1/20 0.70
MEN1 O00255 4/20 0.65
KMT2A Q03164 4/20 0.65
KDM4E B2RXH2 3/20 0.65
MAPT P10636 3/20 0.65
LMNA P02545 2/20 0.65
MAPK1 P28482 1/20 0.64
CETP P11597 1/20 0.59
NPC1 O15118 1/20 0.58
TP53 P04637 1/20 0.58
RAB9A P51151 1/20 0.58
HSD17B10 Q99714 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
RXFP1 Q9HBX9 1/20 0.58
HPGD P15428 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16063220 0.83 NPC1 (0.65) POLBALDH1A1MEN1KMT2AKDM4E
SCHEMBL17831066 0.83 LMNA (0.64) POLBALDH1A1MEN1KMT2AKDM4E
SCHEMBL9923070 0.79 HPGD (0.65) POLBALDH1A1MEN1KMT2AMAPT
SCHEMBL14184555 0.79 POLB (0.67) POLBALDH1A1MEN1KMT2AKDM4E
SCHEMBL20941777 0.79 NOTUM (0.70) POLBALDH1A1MAPTMAPK1CETP
SCHEMBL12883303 0.77 MEN1 (0.56) POLBMEN1KMT2AKDM4EMAPT
SCHEMBL19392493 0.77 MAPT (0.57) POLBALDH1A1MEN1KMT2AKDM4E
SCHEMBL3416858 0.77 HPGD (0.62) POLBALDH1A1MEN1KMT2AKDM4E
SCHEMBL2625088 0.77 POLB (0.76) POLBALDH1A1MEN1KMT2AMAPT
SCHEMBL11211388 0.76 SMN1; SMN2 (0.64) POLBMEN1KMT2AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138356-B2 Chemical inhibitors of inhibitors of differentiation Angiogeney, Inc. (US) 2012-03-20 US disclosed
US-20090226422-A1 Chemical Inhibitors of Inhibitors of Differentiation ANGIOGENEX 2009-09-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090226422-A1 Chemical Inhibitors of Inhibitors of Differentiation BRAF, MAPK1, RAF1 POLB 3542/4885ALDH1A1 1860/4885MEN1 3968/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.