SCHEMBL7410000

SCHEMBL7410000

CS(=O)(=O)OCCCC#Cc1ccc(C#N)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 1/20 0.41
USP2 O75604 1/20 0.41
LMNA P02545 1/20 0.41
MMP9 P14780 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
CA1 P00915 3/20 0.36
CA2 P00918 3/20 0.36
CA9 Q16790 2/20 0.36
MAPT P10636 2/20 0.35
TRPV4 Q9HBA0 1/20 0.35
PPARG P37231 1/20 0.34
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34
CYP2A6 P11509 2/20 0.33
FFAR1 O14842 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
PTGS2 P35354 1/20 0.33
MMP2 P08253 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2903095 0.80 MAPT (0.51) ALDH1A1KDM4EUSP2LMNAMMP9
SCHEMBL7959199 0.80 ALDH1A1 (0.51) ALDH1A1KDM4EUSP2LMNAMMP9
SCHEMBL3871947 0.79 ACACB (0.39) ALDH1A1KDM4EUSP2LMNAMMP9
SCHEMBL23015043 0.79 ALDH1A1 (0.46) ALDH1A1KDM4EUSP2LMNAMMP9
SCHEMBL7417122 0.78 TSHR (0.47) ALDH1A1KDM4EUSP2LMNAMMP9
SCHEMBL2962876 0.77 TSHR (0.50) ALDH1A1KDM4EUSP2LMNAMMP9
SCHEMBL21623467 0.76 CYP2A6 (0.43) ALDH1A1TSHRCA1CA2CA9
SCHEMBL21623418 0.76 CYP2A6 (0.43) ALDH1A1TSHRCA1CA2CA9
SCHEMBL11477234 0.75 PTPN2 (0.37) ALDH1A1KDM4EUSP2LMNAMMP9
SCHEMBL25270396 0.75 HDAC1 (0.56) ALDH1A1KDM4EMMP9MAPTMMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5552431-A ANTICOAGULANTS G. D. SEARLE & CO. (US) 1996-09-03 US disclosed
US-5424334-A Peptide mimetic compounds useful as platelet aggregation inhibitors G. D. SEARLE & CO. (US) 1995-06-13 US disclosed
WO-1993012074-A1 PEPTIDE MIMETIC COMPOUNDS USEFUL AS PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1993-06-24 WO disclosed