SCHEMBL7410015

SCHEMBL7410015

NC(=O)c1cccc2c1OC=CN=C2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 4/20 0.50
PARP1 P09874 10/20 0.41
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
PLK4 O00444 1/20 0.33
CHEK1 O14757 1/20 0.33
AURKA O14965 1/20 0.33
DAPK3 O43293 1/20 0.33
MAP4K4 O95819 1/20 0.33
CSF1R P07333 1/20 0.33
RET P07949 1/20 0.33
FGFR1 P11362 1/20 0.33
PDGFRA P16234 1/20 0.33
LTK P29376 1/20 0.33
KDR P35968 1/20 0.33
MAP2K2 P36507 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2724307 0.84 TRPA1 (0.35) TRPA1ALDH1A1
SCHEMBL7335586 0.74 PARP1 (0.42) TRPA1PARP1KDM4EALDH1A1MAPT
SCHEMBL17766590 0.69 PARP1 (0.47) TRPA1PARP1KDM4EALDH1A1MAPT
SCHEMBL13098173 0.67 TRPA1 (1.00) TRPA1PARP1MAPT
SCHEMBL22612514 0.66 PARP1 (0.44) TRPA1PARP1KDM4EALDH1A1MAPT
SCHEMBL29501123 0.66 TSHR (0.42) PARP1KDM4EALDH1A1TSHRHSD17B10
SCHEMBL29501144 0.66 PIM1 (0.34) ALDH1A1
SCHEMBL7379312 0.65 PARP1 (0.42) TRPA1PARP1KDM4EALDH1A1MAPT
SCHEMBL5322268 0.65 PARP1 (0.54) TRPA1PARP1KDM4EALDH1A1MAPT
SCHEMBL13098214 0.63 TRPA1 (1.00) TRPA1PARP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4935511-A Nervous system, gastrointestinal disorders RORER PHARMACEUTICAL CORPORATION (US) 1990-06-19 US disclosed