SCHEMBL7410253

SCHEMBL7410253

CCCN1CCCC(c2nc3c(OC(N)=O)c(C(C)C)ccc3[nH]2)C1

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 16/20 0.57
PARP2 Q9UGN5 2/20 0.48
ACHE P22303 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7421139 0.95 PARP1 (0.60) PARP1PARP2
SCHEMBL7413860 0.90 PARP1 (0.60) PARP1PARP2
SCHEMBL6864930 0.81 PARP1 (0.65) PARP1PARP2
SCHEMBL7411210 0.79 PARP1 (0.37) PARP1PARP2
SCHEMBL7410717 0.79 PARP1 (0.39) PARP1PARP2
SCHEMBL5621048 0.76 PARP1 (0.88) PARP1PARP2
SCHEMBL6873574 0.76 PARP1 (0.73) PARP1PARP2
Hydrochloric Acid SCHEMBL18614331 0.76 PARP1 (0.86) PARP1PARP2
SCHEMBL7410700 0.74 PARP1 (0.57) PARP1PARP2
SCHEMBL7417789 0.72 PARP1 (0.63) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed