SCHEMBL7410317

SCHEMBL7410317

COc1cc(C#N)c(CCCCC(=O)O)c(C#N)c1O

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 2/20 0.40
STING1 Q86WV6 1/20 0.40
S1PR1 P21453 2/20 0.39
ERBB2 P04626 3/20 0.39
EGFR P00533 2/20 0.39
IMPDH1 P20839 2/20 0.39
HPGD P15428 1/20 0.38
ALOX5 P09917 3/20 0.37
FFAR1 O14842 2/20 0.36
CYP2C9 P11712 1/20 0.36
POLB P06746 1/20 0.36
MAPK1 P28482 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
FFAR4 Q5NUL3 1/20 0.36
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7417930 0.92 STING1 (0.43) IMPDH2STING1S1PR1ERBB2EGFR
SCHEMBL15535456 0.83 TNKS2 (0.48) EGFRALOX5MAPK1TSHR
SCHEMBL7417680 0.83 F13A1 (0.38) IMPDH2IMPDH1HPGDFFAR1SMN1; SMN2
SCHEMBL28817318 0.82 FFAR1 (0.46) S1PR1ALOX5FFAR1FFAR4
SCHEMBL15535114 0.78 GAA (0.46) S1PR1HPGDTSHR
SCHEMBL16978280 0.77 SMN1; SMN2 (0.39) EGFRHPGDALOX5CYP2C9POLB
SCHEMBL15535108 0.76 EGFR (0.36) EGFRHPGDALOX5CYP2C9POLB
SCHEMBL7416187 0.74 FFAR1 (0.38) IMPDH2HPGDFFAR1FFAR4
SCHEMBL16969026 0.73 ERN1 (0.43) HPGD
SCHEMBL15534789 0.73 KDM4E (0.43) ALOX5SMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6150412-A SUCH AS 4-(5-HYDROXY-4-METHOXY-2-NITROPHENYL)BUTANOIC ACID; ADMINISTERING TO INHIBIT CATECHOL-O-METHYL TRANSFERASE; TREATING PARKINSON'S DISEASE OR HYPERTENSION ORION-YHTYMA OY (FI) 2000-11-21 US disclosed
WO-1996037456-A1 NEW CATECHOL DERIVATIVES Orion-Yhtymä Oy (FI) 1996-11-28 WO disclosed