SCHEMBL7417680

SCHEMBL7417680

N#Cc1cc(O)c(O)c(C#N)c1CCCCC(=O)O

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
F13A1 P00488 3/20 0.38
FFAR1 O14842 4/20 0.37
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GLA P06280 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
MAPT P10636 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
FFAR4 Q5NUL3 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
KDM5B Q9UGL1 2/20 0.33
IMPDH2 P12268 1/20 0.33
KDM4A O75164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
IMPDH1 P20839 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7416187 0.91 FFAR1 (0.38) FFAR1KDM4EALDH1A1GLAGAA
SCHEMBL7410317 0.83 IMPDH2 (0.40) FFAR1HPGDFFAR4SMN1; SMN2IMPDH2
SCHEMBL15534992 0.80 KDM4E (0.36) KDM4EMAPT
SCHEMBL11033418 0.75 F13A1 (0.40) F13A1FFAR1MAPTRXFP1HSD17B10
SCHEMBL15535458 0.75 RXRA (0.43) FFAR1KDM4EALDH1A1GAAHPGD
SCHEMBL7417930 0.73 STING1 (0.43) FFAR1ALDH1A1HPGDFFAR4KDM5B
SCHEMBL16969037 0.73 FFAR1 (0.45) FFAR1FFAR4
SCHEMBL15535460 0.72 ESR1 (0.32)
SCHEMBL15535802 0.72 ESR1 (0.36) KDM4EALDH1A1GAAHPGDMAPT
SCHEMBL10763138 0.71 KMO (0.36) F13A1FFAR1FFAR4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6150412-A SUCH AS 4-(5-HYDROXY-4-METHOXY-2-NITROPHENYL)BUTANOIC ACID; ADMINISTERING TO INHIBIT CATECHOL-O-METHYL TRANSFERASE; TREATING PARKINSON'S DISEASE OR HYPERTENSION ORION-YHTYMA OY (FI) 2000-11-21 US disclosed
WO-1996037456-A1 NEW CATECHOL DERIVATIVES Orion-Yhtymä Oy (FI) 1996-11-28 WO disclosed