SCHEMBL7411990

SCHEMBL7411990

COc1ccccc1CC(NN(C(=O)OC(C)(C)C)[C@@H](Cc1ccccc1)C(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 2/20 0.59
ITGB7 P26010 2/20 0.59
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
TACR1 P25103 1/20 0.42
OPRK1 P41145 5/20 0.41
ACE P12821 2/20 0.39
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
FPR2 P25090 1/20 0.38
CACNA1B Q00975 1/20 0.38
KLK5 Q9Y337 1/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7445887 1.00 ITGA4 (0.59) ITGA4ITGB7ALDH1A1GAATACR1
SCHEMBL2386586 0.96 ITGA4 (0.56) ITGA4ITGB7ALDH1A1GAATACR1
SCHEMBL7389438 0.94 ITGA4 (0.55) ITGA4ITGB7ALDH1A1GAATACR1
SCHEMBL2386899 0.93 ITGA4 (0.53) ITGA4ITGB7ALDH1A1GAATACR1
SCHEMBL2387711 0.87 ITGA4 (0.48) ITGA4ITGB7ALDH1A1GAATACR1
SCHEMBL2385811 0.87 ITGA4 (0.46) ITGA4ITGB7ALDH1A1GAAMEN1
SCHEMBL2387173 0.87 ITGA4 (0.48) ITGA4ITGB7ALDH1A1GAATACR1
SCHEMBL2385485 0.86 ITGA4 (0.49) ITGA4ITGB7ALDH1A1ACEMEN1
SCHEMBL2386839 0.86 ITGA4 (0.47) ITGA4ITGB7ALDH1A1GAAACE
SCHEMBL2386831 0.85 ITGA4 (0.47) ITGA4ITGB7ALDH1A1GAATACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6191171-B1 ANTAGONISTS, USEFUL IN INHIBITION OR PREVENTION OF CELL ADHESION AND CELL-ADHESION MEDIATED PATHOLOGIES; FOR DRUGS FOR TREATMENT OF ASTHMA, ALLERGIES, INFLAMMATION, MULTIPLE SCLEROSIS, AND OTHER INFLAMMATORY AND AUTOIMMUNE DISORDERS MERCK & CO., INC. 2001-02-20 US disclosed
WO-1999026923-A1 PARA-AMINOMETHYLARYL CARBOXAMIDE DERIVATIVES MERCK & CO., INC. (US) 1999-06-03 WO disclosed