SCHEMBL7412229

SCHEMBL7412229

CC(=O)c1ccc(-c2ccc(C(C)C(=O)O)cc2F)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 9/20 0.74
AKR1C2 P52895 9/20 0.74
PTGS2 P35354 4/20 0.74
PTGS1 P23219 3/20 0.74
CYP2C19 P33261 3/20 0.74
MEN1 O00255 2/20 0.74
KMT2A Q03164 2/20 0.74
CYP2C9 P11712 2/20 0.74
PSEN1 P49768 2/20 0.74
PSEN2 P49810 2/20 0.74
APH1B Q8WW43 2/20 0.74
NCSTN Q92542 2/20 0.74
APH1A Q96BI3 2/20 0.74
PSENEN Q9NZ42 2/20 0.74
FABP2 P12104 1/20 0.74
TSHR P16473 1/20 0.74
AKR1C4 P17516 1/20 0.74
ADRA2B P18089 1/20 0.74
CHRM3 P20309 1/20 0.74
HTR2C P28335 1/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9667811 0.87 AKR1C3 (0.80) AKR1C3AKR1C2PTGS2PTGS1CYP2C19
4'-Hydroxyflurbiprofen SCHEMBL7040151 0.85 APP (0.97) AKR1C3AKR1C2PTGS2PTGS1CYP2C19
4'-Hydroxyflurbiprofen SCHEMBL6450842 0.85 APP (0.97) AKR1C3AKR1C2PTGS2PTGS1CYP2C19
Flurbiprofen SCHEMBL28766226 0.85 AKR1C3 (0.94) AKR1C3AKR1C2PTGS2PTGS1CYP2C19
Tarenflurbil SCHEMBL26131 0.85 AKR1C3 (1.00) AKR1C3AKR1C2PTGS2PTGS1CYP2C19
Flurbiprofen SCHEMBL8755275 0.85 AKR1C3 (1.00) AKR1C3AKR1C2PTGS2PTGS1CYP2C19
Flurbiprofen SCHEMBL8754830 0.85 AKR1C3 (1.00) AKR1C3AKR1C2PTGS2PTGS1CYP2C19
Esflurbiprofen SCHEMBL505817 0.85 AKR1C3 (1.00) AKR1C3AKR1C2PTGS2PTGS1CYP2C19
Flurbiprofen SCHEMBL10029029 0.85 AKR1C3 (1.00) AKR1C3AKR1C2PTGS2PTGS1CYP2C19
Flurbiprofen SCHEMBL8754978 0.85 AKR1C3 (1.00) AKR1C3AKR1C2PTGS2PTGS1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979226-A1 ISOXAZOLE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2000-02-16 EP disclosed
WO-1998047880-A1 ISOXAZOLE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1998-10-29 WO disclosed
EP-0511021-A1 Novel thiazole derivatives SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1992-10-28 EP disclosed