SCHEMBL7412288

SCHEMBL7412288

COc1ccc(Br)cc1S(=O)(=O)N[C@@H](Cc1ccc(OCCCONC(=N)N)cc1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 14/20 0.48
ITGA2B P08514 11/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C19 P33261 1/20 0.48
ITGAV P06756 3/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
PPARG P37231 1/20 0.42
MMP2 P08253 1/20 0.41
MMP9 P14780 1/20 0.41
GLA P06280 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL7414775 0.96 CYP3A4 (0.47) ITGB3ITGA2BCYP3A4CYP2C19ITGAV
SCHEMBL7421961 0.92 ITGB3 (0.53) ITGB3ITGA2BCYP3A4CYP2C19ITGAV
SCHEMBL7695352 0.91 ITGB3 (0.49) ITGB3ITGA2BCYP3A4CYP2C19ITGAV
SCHEMBL7411729 0.90 ITGB3 (0.53) ITGB3ITGA2BCYP3A4CYP2C19ITGAV
Trifluoroacetic Acid SCHEMBL7415172 0.88 ITGB3 (0.50) ITGB3ITGA2BCYP3A4CYP2C19ITGAV
SCHEMBL7414225 0.88 ITGB3 (0.50) ITGB3ITGA2BMEN1KMT2APPARG
SCHEMBL7414783 0.88 CYP3A4 (0.43) ITGB3ITGA2BCYP3A4CYP2C19ITGAV
SCHEMBL7695459 0.87 ITGB3 (0.49) ITGB3ITGA2BITGAVMEN1KMT2A
Trifluoroacetic Acid SCHEMBL7419764 0.87 CYP3A4 (0.47) ITGB3ITGA2BCYP3A4CYP2C19ITGAV
Trifluoroacetic Acid SCHEMBL7418891 0.86 ITGB3 (0.49) ITGB3ITGA2BCYP3A4CYP2C19ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US claimed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP claimed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO claimed