SCHEMBL7412932

SCHEMBL7412932

CC(C)(C)OC(=O)N=C(NOCCCOc1ccc(C[C@H](N)C(=O)OC(C)(C)C)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 4/20 0.42
ITGA2B P08514 4/20 0.42
CA1 P00915 7/20 0.37
CA2 P00918 7/20 0.37
CA12 O43570 5/20 0.37
CA9 Q16790 5/20 0.37
LTA4H P09960 1/20 0.37
SUCNR1 Q9BXA5 4/20 0.35
PPARG P37231 1/20 0.34
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34
ACACB O00763 1/20 0.34
BCL2 P10415 1/20 0.34
HDAC8 Q9BY41 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7417687 0.88 ITGB3 (0.43) ITGB3ITGA2BCA1CA2CA12
SCHEMBL7408405 0.83 ITGB3 (0.53) ITGB3ITGA2BBCL2
SCHEMBL7407517 0.82 ITGB3 (0.50) ITGB3ITGA2BCA1CA2CA12
SCHEMBL1541948 0.78 ITGB3 (0.59) ITGB3ITGA2BCA1CA2CA12
SCHEMBL16940459 0.77 ITGB3 (0.51) ITGB3ITGA2BLTA4HACACB
SCHEMBL30149840 0.76 CA12 (0.60) ITGB3ITGA2BCA1CA2CA12
SCHEMBL6871466 0.74 ITGB3 (0.51) ITGB3ITGA2BLTA4HPPARG
SCHEMBL7358634 0.73 ACACB (0.50) ITGB3ITGA2BLTA4HPPARGPPARD
SCHEMBL14131858 0.73 CA1 (0.33) CA1CA2CA12CA9
SCHEMBL15149719 0.73 CA12 (0.42) ITGB3ITGA2BCA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6344484-B1 TREATMENT OF TUMOR GROWTH, METASTASIS, OSTEOPOROSIS, RESTENOSIS, INFLAMMATION, MACULAR DEGENERATION, DIABETIC RETINOPATHY, AND RHEUMATOID ARTHRITIS 3-DIMENSIONAL PHARMACEUTICALS, INC. 2002-02-05 US disclosed
EP-1159262-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-12-05 EP disclosed
WO-2000047552-A1 TYROSINE ALKOXYGUANIDINES AS INTEGRIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2000-08-17 WO disclosed