SCHEMBL7413003

SCHEMBL7413003

COC(=O)Cc1cccc(Br)c1.O=C(O)Cc1cccc(Br)c1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 1/20 0.54
EGFR P00533 3/20 0.49
ERBB2 P04626 3/20 0.49
GLA P06280 1/20 0.46
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45
GFER P55789 1/20 0.45
KDM4E B2RXH2 1/20 0.45
FFAR1 O14842 2/20 0.45
FFAR4 Q5NUL3 2/20 0.45
HSP90AB1 P08238 1/20 0.45
HCAR2 Q8TDS4 1/20 0.44
PTGDR2 Q9Y5Y4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL136054 0.94 SLC7A5 (0.55) SLC7A5EGFRERBB2GLAALDH1A1
SCHEMBL29700723 0.94 SLC7A5 (0.55) SLC7A5EGFRERBB2GLAALDH1A1
SCHEMBL1560308 0.89 SLC7A5 (0.65) SLC7A5ALDH1A1GAAGFERKDM4E
SCHEMBL3421266 0.88 SLC7A5 (0.54) SLC7A5EGFRERBB2ALDH1A1GAA
SCHEMBL78652 0.87 AKR1B1 (0.58) EGFRERBB2GAAKDM4EFFAR1
Methane SCHEMBL10697726 0.85 AKR1B1 (0.56) EGFRERBB2GAAKDM4EFFAR1
Hydrochloric Acid SCHEMBL1374336 0.85 AKR1B1 (0.56) EGFRERBB2GAAKDM4EFFAR1
SCHEMBL30267713 0.83 EGFR (0.47) SLC7A5EGFRERBB2GLAKDM4E
SCHEMBL17111341 0.83 EGFR (0.47) SLC7A5EGFRERBB2GLAKDM4E
SCHEMBL12400239 0.81 SLC7A5 (0.68) SLC7A5ALDH1A1GAAGFERKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1079821-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2001-08-29 EP disclosed
EP-1079821-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-03-07 EP disclosed
WO-1999059570-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1999-11-25 WO disclosed