SCHEMBL7413446

SCHEMBL7413446

N#CCCC(C#N)(CCC#N)c1ccc(OC(F)F)c(OCC2CC2)c1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.51
HSD17B10 Q99714 1/20 0.51
PDE4B Q07343 15/20 0.45
PDE4D Q08499 11/20 0.45
PDE4A P27815 7/20 0.45
PDE4C Q08493 7/20 0.45
ABCB11 O95342 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28279542 0.86 PDE4B (0.47) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL7866895 0.85 PDE4B (0.49) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL7865357 0.83 PDE4B (0.52) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL25111149 0.77 PDE4B (0.56) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL28242988 0.76 PDE4B (0.52) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL29723277 0.76 PDE4B (0.56) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL16650722 0.76 PDE4B (0.56) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL7421380 0.75 PDE4B (0.51) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL22713890 0.73 PDE4B (0.43) PDE4BPDE4DPDE4APDE4CABCB11
SCHEMBL30352593 0.73 PDE4B (0.43) PDE4BPDE4DPDE4APDE4CABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5449687-A 4-phenyl-1,2-cyclohexyl derivatives and anti-inflammatory compositions and methods thereof SMITHKLINE BEECHAM CORPORATION (US) 1995-09-12 US disclosed
EP-0633771-A4 COMPOUNDS. 1995-02-22 EP disclosed
EP-0633771-A1 COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1995-01-18 EP disclosed
WO-1993019720-A2 COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1993-10-14 WO disclosed