SCHEMBL741372

SCHEMBL741372

COc1cccc2[nH]c([C@@H]3CCCNC3)nc12

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.61
ADORA2A P29274 1/20 0.50
HTR2A P28223 9/20 0.46
PARP2 Q9UGN5 2/20 0.43
HTR2C P28335 4/20 0.42
IKBKB O14920 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741373 1.00 PARP1 (0.61) PARP1ADORA2AHTR2APARP2HTR2C
SCHEMBL30689173 0.87 PARP1 (0.56) PARP1ADORA2APARP2HTR2C
SCHEMBL27041996 0.87 PARP1 (0.56) PARP1ADORA2APARP2HTR2C
SCHEMBL5201219 0.84 PARP1 (0.55) PARP1ADORA2APARP2
SCHEMBL742068 0.83 PARP1 (0.65) PARP1PARP2
SCHEMBL742067 0.83 PARP1 (0.65) PARP1PARP2
SCHEMBL6864453 0.82 PARP1 (0.71) PARP1PARP2
SCHEMBL14587803 0.81 PARP1 (0.65) PARP1HTR2APARP2HTR2C
Hydrochloric Acid SCHEMBL4716384 0.80 PARP1 (0.63) PARP1HTR2APARP2HTR2C
SCHEMBL762835 0.78 PARP1 (0.64) PARP1HTR2APARP2HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed