SCHEMBL762835

SCHEMBL762835

COc1cccc2[nH]c([C@@H]3CCCN(C)C3)nc12

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.64
PARP2 Q9UGN5 1/20 0.45
HCRTR1 O43613 2/20 0.45
HCRTR2 O43614 2/20 0.45
POLB P06746 1/20 0.43
DRD2 P14416 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
KCNH2 Q12809 1/20 0.43
CCNT1 O60563 2/20 0.42
CDK9 P50750 2/20 0.42
PDE10A Q9Y233 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6872852 0.85 PARP1 (0.72) PARP1PARP2
SCHEMBL30096832 0.83 PARP1 (0.49) PARP1POLBDRD2HTR2AHTR2C
SCHEMBL5201219 0.82 PARP1 (0.55) PARP1PARP2HCRTR1HCRTR2POLB
SCHEMBL741850 0.80 PARP1 (0.51) PARP1HCRTR1HCRTR2POLB
SCHEMBL741851 0.80 PARP1 (0.51) PARP1HCRTR1HCRTR2POLB
SCHEMBL5621503 0.78 PARP1 (1.00) PARP1PARP2
SCHEMBL741373 0.78 PARP1 (0.61) PARP1PARP2HTR2AHTR2C
SCHEMBL741372 0.78 PARP1 (0.61) PARP1PARP2HTR2AHTR2C
Hydrochloric Acid SCHEMBL18614328 0.77 PARP1 (0.98) PARP1PARP2
SCHEMBL16349536 0.77 PARP1 (0.59) PARP1POLBDRD2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed