SCHEMBL7414308

SCHEMBL7414308

Cc1cccc2c1Oc1ccc(Cl)cc1N=C2N1CCN(C)CC1

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 12/20 0.82
DRD2 P14416 7/20 0.71
DRD4 P21917 6/20 0.71
ADRA2A P08913 4/20 0.66
HTR2A P28223 4/20 0.66
DRD1 P21728 5/20 0.61
HRH2 P25021 3/20 0.61
HRH1 P35367 3/20 0.61
ADRB2 P07550 2/20 0.61
CHRM2 P08172 2/20 0.61
CHRM4 P08173 2/20 0.61
HTR1A P08908 2/20 0.61
CHRM5 P08912 2/20 0.61
CHRM1 P11229 2/20 0.61
ADRA2B P18089 2/20 0.61
ADRA2C P18825 2/20 0.61
CHRM3 P20309 2/20 0.61
TBXA2R P21731 2/20 0.61
DRD5 P21918 2/20 0.61
SLC6A2 P23975 2/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7404974 0.92 HRH4 (0.82) HRH4DRD2DRD4ADRA2AHTR2A
SCHEMBL7404036 0.90 HRH4 (0.85) HRH4DRD2DRD4ADRA2AHTR2A
SCHEMBL3408030 0.88 HTR2A (0.65) HRH4DRD2DRD4ADRA2AHTR2A
Isoloxapine SCHEMBL2738975 0.83 HRH4 (1.00) HRH4DRD2DRD4ADRA2AHTR2A
SCHEMBL7410631 0.82 HRH4 (0.84) HRH4DRD2DRD4ADRA2AHTR2A
SCHEMBL3411352 0.80 HRH4 (0.64) HRH4DRD2DRD4ADRA2AHTR2A
SCHEMBL2615392 0.80 HRH4 (0.78) HRH4DRD2DRD4ADRA2AHTR2A
SCHEMBL9216773 0.80 DRD4 (1.00) HRH4DRD2DRD4ADRA2AHTR2A
SCHEMBL11505616 0.79 HRH4 (0.74) HRH4DRD2DRD4ADRA2AHTR2A
SCHEMBL15963179 0.77 HRH4 (0.75) HRH4DRD2DRD4ADRA2AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3962248-A PROCESS FOR MAKING 11-PIPERAZINO-DIAZEPINES, OXAZEPINES, THIAZEPINES AND AZEPINES SANDOZ, INC. (US) 1976-06-08 US disclosed