SCHEMBL7414719

SCHEMBL7414719

ClCCCSc1ccc(Cl)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.54
HDAC4 P56524 1/20 0.54
HDAC1 Q13547 1/20 0.54
HDAC7 Q8WUI4 1/20 0.54
HDAC2 Q92769 1/20 0.54
HDAC10 Q969S8 1/20 0.54
HDAC11 Q96DB2 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
HDAC9 Q9UKV0 1/20 0.54
HDAC5 Q9UQL6 1/20 0.54
KDM4E B2RXH2 7/20 0.50
ALDH1A1 P00352 6/20 0.50
TEAD1 P28347 1/20 0.50
YAP1 P46937 1/20 0.50
TEAD4 Q15561 1/20 0.50
TEAD2 Q15562 1/20 0.50
PKM P14618 1/20 0.50
DRD2 P14416 3/20 0.47
MEN1 O00255 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10917708 0.93 KDM4E (0.53) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL9808024 0.88 KDM4E (0.59) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL9808069 0.88 KDM4E (0.55) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL1274257 0.86 TEAD1 (0.53) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL9808062 0.83 TEAD1 (0.53) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL3908789 0.82 CYP2A6 (0.42) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL9493058 0.81 KDM4E (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL9580278 0.81 HDAC3 (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4025742 0.81 HDAC3 (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7009525 0.81 HDAC3 (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1671386-A Substituted anilinic piperidines as MCH selective antagonists LUNDBECK & CO AS H (DK) 2005-09-21 CN disclosed
EP-0393574-B1 Hexitol derivatives KYOWA HAKKO KOGYO KK (JP) 1996-01-31 EP disclosed
US-5198449-A N-substituted alpha-arylazacycloalkylmethanamines and their use as cardiovascular agents A. H. ROBINS COMPANY INCORPORATED (US) 1993-03-30 US disclosed
US-5053408-A Cardiovascular disorders KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-10-01 US disclosed
EP-0393574-A2 Hexitol derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1990-10-24 EP disclosed
EP-0001654-B1 IMIDAZOLYLETHYLENE-OXYALKYLOXY DERIVATIVES AND THEIR THIO ANALOGUES, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SIEGFRIED AKTIENGESELLSCHAFT (CH) 1981-07-22 EP disclosed
US-4177350-A FUNGICIDES SIEGFRIED AKTIENGESELLSCHAFT (CH) 1979-12-04 US disclosed
EP-0001654-A1 Imidazolylethylene-oxyalkyloxy derivatives and their thio analogues, methods for their preparation and pharmaceutical compositions containing them SIEGFRIED AKTIENGESELLSCHAFT (CH) 1979-05-02 EP disclosed