SCHEMBL7414784

SCHEMBL7414784

BrC1=CC=Cc2ccccc2N1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.54
GAA P10253 1/20 0.54
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
P2RX4 Q99571 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31188758 1.00 MAPT (0.54) MAPTGAARAB9ASMN1; SMN2P2RX4
SCHEMBL29605097 0.75 MAPT (0.54) MAPTGAARAB9ASMN1; SMN2P2RX4
SCHEMBL30823596 0.75 MAPT (0.54) MAPTGAARAB9ASMN1; SMN2P2RX4
SCHEMBL30462264 0.75 MAPT (0.54) MAPTGAARAB9ASMN1; SMN2P2RX4
SCHEMBL9935617 0.75 MAPT (0.54) MAPTGAARAB9ASMN1; SMN2P2RX4
SCHEMBL31482354 0.75 MAPT (0.54) MAPTGAARAB9ASMN1; SMN2P2RX4
SCHEMBL8769697 0.75 MAPT (0.54) MAPTGAARAB9ASMN1; SMN2P2RX4
SCHEMBL29181630 0.75 MAPT (0.54) MAPTGAARAB9ASMN1; SMN2P2RX4
SCHEMBL460837 0.75 MAPT (0.54) MAPTGAARAB9ASMN1; SMN2P2RX4
SCHEMBL6312855 0.75 MAPT (0.54) MAPTGAARAB9ASMN1; SMN2P2RX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119059958-A Method for aryl debromination acylation of bromobenzazepine compounds 上海沃凯生物技术有限公司 2024-12-03 CN claimed
CN-119059958-A Method for aryl debromination acylation of bromobenzazepine compounds 上海沃凯生物技术有限公司 2024-12-03 CN disclosed
CN-119059958-A Method for aryl debromination acylation of bromobenzazepine compounds 上海沃凯生物技术有限公司 2024-12-03 CN disclosed
CN-119059958-A Method for aryl debromination acylation of bromobenzazepine compounds 上海沃凯生物技术有限公司 2024-12-03 CN disclosed
CN-115286566-B Synthesis method of pheniramine or derivatives thereof 南京农业大学 2023-09-19 CN disclosed
CN-116368168-A Novel antimicrobial and antithrombotic medical device 列日大学 2023-06-30 CN disclosed
CN-106164044-B Process for producing 1-arylimino-2-vinylcyclopropanecarboxylic acid derivative 株式会社钟化 2018-05-04 CN disclosed
CN-106164044-A Process for producing 1-arylimino-2-vinylcyclopropanecarboxylic acid derivative 株式会社钟化 2016-11-23 CN disclosed
CN-1859949-A New derivative of 4A,5,9,10,11,12-tetrahydro-6H-benzofuro[3A, 3, 2-EF] [2] benzazepinium bromide, method of preparation thereof and use in the production of medicaments SANOCHEMIA PHARMAZEUTIKA AG (AT) 2006-11-08 CN disclosed
US-5063230-A Substituted saturated and unsaturated indole quinoline and benzazepine carboxamides and their use as pharmacological agents RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-11-05 US disclosed
WO-1990006113-A1 SUBSTITUTED SATURATED AND UNSATURATED INDOLE QUINOLINE AND BENZAZEPINE CARBOXAMIDES AND THEIR USE AS PHARMACOLOGICAL AGENTS RORER INTERNATIONAL (OVERSEAS) INC. (US) 1990-06-14 WO disclosed
EP-0230755-B1 1-PHENYL-3-BENZAZEPINES SMITHKLINE BEECHAM CORPORATION (US) 1990-05-16 EP disclosed
US-4920219-A Substituted saturated and unsaturated indole quinoline and benzazepine carboxamides and their use as pharmacological agents RORER PHARMACEUTICAL CORP. (US) 1990-04-24 US disclosed
US-4707483-A 1-phenyl-3-benzazepines and their use for treating gastrointestinal motility disorders SMITHKLINE BECKMAN CORPORATION (US) 1987-11-17 US disclosed
EP-0230755-A1 1-Phenyl-3-benzazepines SMITHKLINE BEECHAM CORPORATION (US) 1987-08-05 EP disclosed