SCHEMBL7414824

SCHEMBL7414824

CC(Cl)CC(=O)c1ccc2c(c1)CC(=O)N2

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.56
SMYD3 Q9H7B4 16/20 0.52
AHR P35869 1/20 0.48
HTR1A P08908 1/20 0.47
DRD2 P14416 1/20 0.47
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
HTR7 P34969 1/20 0.47
DRD3 P35462 1/20 0.47
HTR2B P41595 1/20 0.47
GRIN2B Q13224 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5774940 0.89 EPHX2 (0.58) EPHX2SMYD3AHRHTR1ADRD2
Hydrochloric Acid SCHEMBL8141533 0.86 EPHX2 (0.56) EPHX2SMYD3HTR1ADRD2HTR2A
SCHEMBL7985233 0.82 SMYD3 (0.52) EPHX2SMYD3AHR
SCHEMBL1304506 0.81 EPHX2 (0.59) EPHX2SMYD3AHRHTR1ADRD2
SCHEMBL4304359 0.81 EPHX2 (0.62) EPHX2SMYD3AHRHTR1ADRD2
SCHEMBL3389331 0.80 EPHX2 (0.61) EPHX2SMYD3AHRHTR1ADRD2
SCHEMBL6225349 0.80 EPHX2 (0.57) EPHX2SMYD3AHRHTR1ADRD2
Hydrochloric Acid SCHEMBL7036110 0.79 EPHX2 (0.56) EPHX2SMYD3AHRHTR1ADRD2
Hydrochloric Acid SCHEMBL7036109 0.79 EPHX2 (0.56) EPHX2SMYD3AHRHTR1ADRD2
SCHEMBL1557916 0.79 SMYD3 (0.54) EPHX2SMYD3AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0281309-B1 PIPERAZINYL-HETEROCYCLIC COMPOUNDS PFIZER INC. (US) 1991-12-27 EP disclosed
US-4883795-A Piperazinyl-heterocyclic compounds PFIZER INC. (US) 1989-11-28 US disclosed
US-4831031-A Aryl piperazinyl-(C2 or C4) alkylene heterocyclic compounds having neuroleptic activity PFIZER INC. (US) 1989-05-16 US disclosed
EP-0281309-A1 Piperazinyl-heterocyclic compounds PFIZER INC. (US) 1988-09-07 EP disclosed