SCHEMBL741582

SCHEMBL741582

COCCCn1c(C2CCCN(C(=O)CC(N)c3cccc(Cl)c3)C2)nc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.44
MAPT P10636 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KCNH2 Q12809 8/20 0.44
HRH1 P35367 10/20 0.44
CYP2D6 P10635 6/20 0.44
CHRM1 P11229 3/20 0.44
PROKR1 Q8TCW9 1/20 0.40
USP2 O75604 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL741581 1.00 TP53 (0.44) TP53MAPTSMN1; SMN2KCNH2HRH1
SCHEMBL741047 0.91 HRH1 (0.50) KCNH2HRH1CYP2D6CHRM1USP2
SCHEMBL739699 0.91 HRH1 (0.50) KCNH2HRH1CYP2D6CHRM1USP2
SCHEMBL741011 0.91 HRH1 (0.50) KCNH2HRH1CYP2D6CHRM1USP2
SCHEMBL741010 0.91 HRH1 (0.50) KCNH2HRH1CYP2D6CHRM1USP2
SCHEMBL742589 0.91 KCNH2 (0.48) TP53MAPTSMN1; SMN2KCNH2HRH1
SCHEMBL762869 0.91 KCNH2 (0.48) TP53MAPTSMN1; SMN2KCNH2HRH1
SCHEMBL739630 0.91 KCNH2 (0.44) KCNH2HRH1CYP2D6CHRM1PROKR1
SCHEMBL739631 0.91 KCNH2 (0.44) KCNH2HRH1CYP2D6CHRM1PROKR1
SCHEMBL741491 0.89 HRH1 (0.42) KCNH2HRH1CYP2D6CHRM1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US claimed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed