SCHEMBL7416050

SCHEMBL7416050

Cc1c(Cl)c[nH]c(=O)c1Br

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DAO P14920 4/20 0.33
HPGD P15428 1/20 0.33
ADRA1A P35348 1/20 0.33
ERCC1 P07992 1/20 0.33
ERCC4 Q92889 1/20 0.33
GRIN2D O15399 2/20 0.32
GRIN3B O60391 2/20 0.32
GRIN1 Q05586 2/20 0.32
GRIN2A Q12879 2/20 0.32
GRIN2B Q13224 2/20 0.32
GRIN2C Q14957 2/20 0.32
GRIN3A Q8TCU5 2/20 0.32
ATAD2 Q6PL18 1/20 0.31
DYRK1A Q13627 1/20 0.31
CSNK2A2 P19784 1/20 0.30
CSNK2B P67870 1/20 0.30
CSNK2A1 P68400 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7422492 0.77 DAO (0.35) DAOHPGDERCC1ERCC4ATAD2
SCHEMBL16976171 0.77 ATAD2 (0.43) DAOHPGDERCC1ERCC4GRIN2D
SCHEMBL27295589 0.74 ERCC1 (0.34) DAOADRA1AERCC1ERCC4GRIN2D
SCHEMBL27791441 0.73 DAO (0.35) DAOHPGDADRA1AGRIN2DGRIN3B
SCHEMBL16654409 0.70 DAO (0.33) DAOERCC1ERCC4GRIN2DGRIN3B
SCHEMBL1200250 0.68 KDM4E (0.53) HPGDGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL16795068 0.66
SCHEMBL2124039 0.65 DAO (0.37) DAOHPGDERCC1ERCC4GRIN2D
SCHEMBL6292566 0.65 TYMP (0.49) DAO
SCHEMBL30884517 0.64 DAO (0.39) DAOHPGDADRA1AERCC1ERCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110997656-B Substituted indole compounds useful as TLR7/8/9 inhibitors 百时美施贵宝公司 2023-04-14 CN disclosed
EP-1244625-A1 4-PYRIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2002-10-02 EP disclosed
WO-2001042215-A1 4-PYRIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2001-06-14 WO disclosed