SCHEMBL7416787

SCHEMBL7416787

CCCS(=O)(=O)NCc1cccnc1

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.55
POLB P06746 1/20 0.55
TBXAS1 P24557 1/20 0.54
CYP1A2 P05177 2/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C19 P33261 2/20 0.51
ALDH1A1 P00352 2/20 0.50
NPSR1 Q6W5P4 1/20 0.50
IDO1 P14902 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
PKM P14618 1/20 0.50
LMNA P02545 1/20 0.50
HPGD P15428 1/20 0.50
HTT P42858 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6733057 0.89 TSHR (0.58) TSHRPOLBCYP1A2CYP2D6CYP2C19
SCHEMBL1837988 0.88 TDP1 (0.53) TSHRPOLBCYP1A2CYP2D6CYP2C19
SCHEMBL7007840 0.88 TDP1 (0.53) TSHRPOLBCYP1A2CYP2D6CYP2C19
SCHEMBL1099625 0.85 TSHR (0.52) TSHRPOLBCYP1A2CYP2D6CYP2C19
SCHEMBL7011029 0.81 NAMPT (0.57) TSHRPOLBCYP1A2CYP2D6CYP2C19
SCHEMBL3597587 0.80 TSHR (0.60) TSHRPOLBCYP1A2CYP2D6CYP2C19
SCHEMBL24990193 0.80 CA2 (0.59) CYP1A2ALDH1A1CYP3A4HTTSMN1; SMN2
Acetic Acid SCHEMBL28216269 0.78 MAPT (0.56) TSHRPOLBCYP1A2CYP2C19CYP3A4
SCHEMBL6562898 0.77 KMT2A (0.45) TSHRALDH1A1SMN1; SMN2
SCHEMBL7534037 0.77 CYP1A2 (0.50) TSHRPOLBCYP1A2CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255735-A2 PYRIDINE DERIVATIVES AS POTENTIATORS OF GLUTAMATE RECEPTORS ELI LILLY AND COMPANY (US) 2002-11-13 EP claimed
WO-2001056990-A2 PYRIDINE DERIVATES AS POTENTIATORS OF GLUTAMATE RECEPTORS ELI LILLY AND COMPANY (US) 2001-08-09 WO claimed