SCHEMBL7416890

SCHEMBL7416890

CC(=O)Cc1ccc2c(n1)CN(C)C(=O)N2C

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
XIAP P98170 2/20 0.50
BIRC2 Q13490 2/20 0.50
BRD4 O60885 1/20 0.31
BRD2 P25440 1/20 0.31
BRD3 Q15059 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7416891 0.77 XIAP (0.41) XIAPBIRC2
SCHEMBL13826643 0.73 XIAP (0.50) XIAPBIRC2BRD4BRD2BRD3
SCHEMBL7414097 0.73 XIAP (0.50) XIAPBIRC2BRD4BRD2BRD3
SCHEMBL7413307 0.71 BRD4 (0.35) XIAPBIRC2BRD4BRD2BRD3
SCHEMBL7473009 0.69 XIAP (0.45) XIAPBIRC2
SCHEMBL13732112 0.69 XIAP (0.52) XIAPBIRC2
Hydrochloric Acid SCHEMBL13733105 0.68 XIAP (0.51) XIAPBIRC2
SCHEMBL13732110 0.67 BIRC2 (1.00) XIAPBIRC2
Hydrochloric Acid SCHEMBL15467022 0.66 BIRC2 (0.98) XIAPBIRC2
SCHEMBL21932324 0.60 XIAP (0.38) XIAPBIRC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5002944-A Compounds having cardiotonic activity RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-03-26 US disclosed
EP-0333727-A1 HETEROCYCLIC SUBSTITUTED BICYCLOUREAS HAVING CARDIOTONIC ACTIVITY RORER INTERNATIONAL (OVERSEAS) INC. (a Delaware corporation) (US) 1989-09-27 EP disclosed
US-4859672-A Pyrido[2,3-d]pyrimidinone and imidazo[4,5-b]pyrimidinone RORER PHARMACEUTICAL CORPORATION (US) 1989-08-22 US disclosed
WO-1988003025-A1 HETEROCYCLIC SUBSTITUTED BICYCLOUREAS HAVING CARDIOTONIC ACTIVITY RORER INTERNATIONAL (OVERSEAS) INC. (US) 1988-05-05 WO disclosed