SCHEMBL7413307

SCHEMBL7413307

CC(=O)Cc1cc2c(cn1)N(C)C(=O)N(C)C2

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.35
BRD2 P25440 1/20 0.35
BRD3 Q15059 1/20 0.35
FGFR4 P22455 1/20 0.32
XIAP P98170 1/20 0.32
BIRC2 Q13490 1/20 0.32
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7416891 0.73 XIAP (0.41) XIAPBIRC2
SCHEMBL7419734 0.73 ENPP1 (0.31) EGFR
SCHEMBL7416890 0.71 XIAP (0.50) BRD4BRD2BRD3XIAPBIRC2
SCHEMBL19508032 0.66 FGFR4 (0.37) BRD4BRD2BRD3FGFR4XIAP
SCHEMBL12081005 0.64 BRD4 (0.50) BRD4BRD2BRD3
SCHEMBL4859534 0.62 BRD4 (0.40) BRD4BRD2BRD3
SCHEMBL5985150 0.62 BRD4 (0.51) BRD4BRD2BRD3
SCHEMBL21932324 0.62 XIAP (0.38) XIAPBIRC2
SCHEMBL8559372 0.61 BRD4 (0.50) BRD4BRD2BRD3XIAPBIRC2
SCHEMBL29209001 0.61 BRD4 (0.53) BRD4BRD2BRD3EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5002944-A Compounds having cardiotonic activity RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-03-26 US disclosed
EP-0333727-A1 HETEROCYCLIC SUBSTITUTED BICYCLOUREAS HAVING CARDIOTONIC ACTIVITY RORER INTERNATIONAL (OVERSEAS) INC. (a Delaware corporation) (US) 1989-09-27 EP disclosed
US-4859672-A Pyrido[2,3-d]pyrimidinone and imidazo[4,5-b]pyrimidinone RORER PHARMACEUTICAL CORPORATION (US) 1989-08-22 US disclosed
WO-1988003025-A1 HETEROCYCLIC SUBSTITUTED BICYCLOUREAS HAVING CARDIOTONIC ACTIVITY RORER INTERNATIONAL (OVERSEAS) INC. (US) 1988-05-05 WO disclosed