SCHEMBL7417286

SCHEMBL7417286

N#CCNC(=O)c1ccc2ccccc2c1Br

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.53
CTSB P07858 2/20 0.44
CTSS P25774 2/20 0.44
CTSV O60911 1/20 0.44
CTSL P07711 1/20 0.44
MAPT P10636 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
NCEH1 Q6PIU2 4/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.41
HDAC8 Q9BY41 2/20 0.41
MMP3 P08254 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9536835 0.82 PLK1 (0.60) EGLN1CTSBCTSSCTSVCTSL
SCHEMBL2322433 0.79 NCEH1 (0.60) EGLN1SMN1; SMN2NCEH1KMT2AALDH1A1
SCHEMBL15505756 0.79 PLK1 (0.64) MAPTSMN1; SMN2NPC1RAB9ANCEH1
SCHEMBL31047578 0.77 NCEH1 (0.57) SMN1; SMN2NCEH1KDM4EALDH1A1GAA
SCHEMBL27713015 0.77 SMN1; SMN2 (0.44) MAPTSMN1; SMN2NPC1RAB9ANCEH1
SCHEMBL31047597 0.77 NCEH1 (0.57) SMN1; SMN2NCEH1KDM4EALDH1A1GAA
SCHEMBL2332306 0.75 EGLN1 (0.60) EGLN1MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL6844201 0.75 KDM4E (0.48) MAPTSMN1; SMN2NPC1RAB9ANCEH1
SCHEMBL7413948 0.73 NCEH1 (0.43) CTSBCTSSCTSVCTSLMAPT
SCHEMBL31520424 0.73 POLB (0.52) MAPTSMN1; SMN2NPC1RAB9ANCEH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1157003-A1 ACYLATED AMINOACETONITRILES AS CYSTEINE PROTEASE INHIBITORS AstraZeneca AB (SE) 2001-11-28 EP disclosed
WO-2000048992-A1 ACYLATED AMINOACETONITRILES AS CYSTEINE PROTEASE INHIBITORS ASTRAZENECA AB (SE) 2000-08-24 WO disclosed