SCHEMBL7417402

SCHEMBL7417402

COC(=O)c1cc(C(=O)OC)n(CCCN)n1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 2/20 0.38
MAPK1 P28482 2/20 0.34
LCK P06239 1/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
SMPD1 P17405 2/20 0.34
CNR1 P21554 2/20 0.34
CNR2 P34972 2/20 0.34
ADORA3 P0DMS8 1/20 0.33
JMJD6 Q6NYC1 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TLR8 Q9NR97 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12532887 0.91 MAPK1 (0.36) KDM4EALDH1A1HPGDHSD17B10MAPK1
SCHEMBL31460072 0.84 KDM4E (0.38) KDM4EALDH1A1HPGDHSD17B10RAB9A
Hydrochloric Acid SCHEMBL31459957 0.83 KDM4E (0.39) KDM4EALDH1A1HPGDHSD17B10RAB9A
SCHEMBL12532886 0.82 MAPKAPK2 (0.40) KDM4EALDH1A1HPGDHSD17B10MAPK1
SCHEMBL31409379 0.81 TP53 (0.42) KDM4EALDH1A1HPGDHSD17B10NPC1
SCHEMBL24928462 0.81 TSHR (0.39) KDM4EALDH1A1HPGDHSD17B10MAPK1
SCHEMBL23115927 0.80 AURKA (0.39) KDM4EALDH1A1HPGDHSD17B10MAPK1
SCHEMBL30860986 0.79 PDE4A (0.39) KDM4EALDH1A1HPGDHSD17B10SMPD1
SCHEMBL171958 0.78 SMPD1 (0.41) SMPD1CNR1CNR2
SCHEMBL20661071 0.75 CYP11B1 (0.36) KDM4EALDH1A1HPGDHSD17B10MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821241-A INHIBIT BINDING OF FIBRINOGEN TO BLOOD PLATELETS, INHIBIT AGGREGATION OF BLOOD PLATELETS, PREVENT OR TREAT THROMBUS OR EMBOLUS FORMATION MERCK & CO., INC. (US) 1998-10-13 US disclosed
WO-1994018981-A1 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1994-09-01 WO disclosed