SCHEMBL7417628

SCHEMBL7417628

O=C1C=C(C#Cc2ccccn2)CCC1

nearest known ligand 0.63

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 6/20 0.60
CYP1A2 P05177 5/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7422525 0.78 GRM5 (0.56) GRM5CYP1A2
SCHEMBL7422531 0.78 GRM5 (0.56) GRM5CYP1A2
SCHEMBL4160148 0.77 GRM5 (0.65) GRM5CYP1A2
SCHEMBL7387265 0.76 GRM5 (0.50) GRM5CYP1A2
SCHEMBL7419526 0.75 GRM5 (0.46) GRM5CYP1A2
SCHEMBL7383590 0.75 ALDH1A1 (0.50) GRM5CYP1A2
SCHEMBL4860119 0.73 GRM5 (0.97) GRM5CYP1A2
SCHEMBL4864474 0.73 GRM5 (0.97) GRM5CYP1A2
SCHEMBL4864468 0.73 GRM5 (0.97) GRM5CYP1A2
SCHEMBL352291 0.73 GRM5 (0.65) GRM5CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214303-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001016121-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF MERCK & CO., INC. (US) 2001-03-08 WO disclosed