SCHEMBL7419004

SCHEMBL7419004

CC(c1cc(C(F)(F)F)cc(C(F)(F)F)c1)S(=O)(=O)C(C)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.40
TACR1 P25103 5/20 0.38
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37
ACP1 P24666 2/20 0.36
PTPN7 P35236 1/20 0.36
PTPN12 Q05209 1/20 0.36
PTPN13 Q12923 1/20 0.36
SSU72 Q9NP77 1/20 0.36
MAPT P10636 1/20 0.36
ALDH1A1 P00352 1/20 0.36
PDE2A O00408 2/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
CYP2D6 P10635 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
TACR3 P29371 1/20 0.35
XPO1 O14980 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL437277 0.77 TACR1 (0.42) CES2TACR1IDO1TDO2MAPT
SCHEMBL14972564 0.75 TACR1 (0.43) TACR1TACR3
SCHEMBL13484088 0.75 TACR1 (0.43) TACR1TACR3
SCHEMBL4528004 0.75 TACR1 (0.43) TACR1TACR3
SCHEMBL18106081 0.75 TACR1 (0.41) CES2TACR1IDO1TDO2MAPT
SCHEMBL17994000 0.75 TACR1 (0.41) CES2TACR1IDO1TDO2MAPT
SCHEMBL13476400 0.75 TACR1 (0.41) CES2TACR1IDO1TDO2MAPT
SCHEMBL20530516 0.74 MAPT (0.41) CES2TACR1ACP1PTPN7PTPN12
SCHEMBL20730205 0.73 TACR1 (0.40) CES2TACR1IDO1TDO2MAPT
SCHEMBL16953807 0.73 TACR1 (0.40) CES2TACR1IDO1TDO2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1112251-A1 AZETIDINE DERIVATIVES, PREPARATION AND MEDICINES CONTAINING THEM Aventis Pharma S.A. (FR) 2001-07-04 EP disclosed
WO-2000015609-A1 AZETIDINE DERIVATIVES, PREPARATION AND MEDICINES CONTAINING THEM AVENTIS PHARMA S.A. (FR) 2000-03-23 WO disclosed