SCHEMBL7419081

SCHEMBL7419081

CC(C)(C)OC(=O)NCCN(CC(N)=O)C(=O)OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.48
IDO1 P14902 1/20 0.47
CCR6 P51684 1/20 0.45
PAX8 Q06710 1/20 0.45
CKS1B P61024 1/20 0.44
SKP1 P63208 1/20 0.44
SKP2 Q13309 1/20 0.44
MAPT P10636 2/20 0.43
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
SIGMAR1 Q99720 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
CTSS P25774 1/20 0.41
TACR1 P25103 1/20 0.41
HTT P42858 1/20 0.41
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12093506 0.92 SYK (0.49) SYKIDO1CCR6PAX8CKS1B
SCHEMBL2685379 0.91 SYK (0.50) SYKIDO1CCR6PAX8CKS1B
SCHEMBL15716592 0.89 SYK (0.55) SYKIDO1CCR6PAX8CKS1B
SCHEMBL2748437 0.88 SYK (0.49) SYKIDO1CCR6PAX8CKS1B
SCHEMBL16490057 0.87 SYK (0.49) SYKIDO1CCR6PAX8CKS1B
SCHEMBL25346745 0.86 CCR6 (0.52) SYKIDO1CCR6PAX8CKS1B
SCHEMBL25970217 0.86 SYK (0.53) SYKIDO1CCR6PAX8CKS1B
SCHEMBL17948 0.85 IDO1 (0.47) SYKIDO1CCR6PAX8CKS1B
SCHEMBL14023844 0.85 SYK (0.45) SYKIDO1CCR6PAX8CKS1B
SCHEMBL17545677 0.85 SYK (0.49) SYKIDO1CCR6PAX8CKS1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5610165-A N-acylpiperidine tachykinin antagonists MERCK & CO., INC. (US) 1997-03-11 US disclosed
WO-1995022525-A1 N-ACYLPIPERIDINE TACHYKININ ANTAGONISTS MERCK & CO., INC. (US) 1995-08-24 WO disclosed
US-5344830-A Anitinflammatory, cardiovascular, analgesic, central nervous system MERCK & CO., INC. (US) 1994-09-06 US disclosed
WO-1994013646-A1 N,N-DIACYLPIPERAZINE TACHYKININ ANTAGONISTS MERCK & CO., INC. (US) 1994-06-23 WO disclosed