SCHEMBL7419786

SCHEMBL7419786

N#Cc1cccc(CN2C(=O)C[C@H](N)C2=O)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.43
SIRT1 Q96EB6 1/20 0.43
TACR1 P25103 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CYP19A1 P11511 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
MAPT P10636 1/20 0.42
GLA P06280 1/20 0.41
ALDH1A1 P00352 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
GAA P10253 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
STAT6 P42226 1/20 0.40
CHRM3 P20309 1/20 0.40
FAAH O00519 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2334099 0.99 SIRT2 (0.42) SIRT2SIRT1TACR1L3MBTL1CYP19A1
Hydrochloric Acid SCHEMBL2334098 0.99 SIRT2 (0.42) SIRT2SIRT1TACR1L3MBTL1CYP19A1
SCHEMBL7419782 0.83 SIRT2 (0.50) SIRT2SIRT1TACR1L3MBTL1CYP19A1
SCHEMBL7427087 0.78 SIRT2 (0.53) SIRT2SIRT1L3MBTL1CYP19A1CYP11B1
SCHEMBL22426223 0.78 ALDH1A1 (0.60) MAPTALDH1A1CYP1A2CYP3A4GAA
SCHEMBL5180380 0.78 ALDH1A1 (0.60) MAPTALDH1A1CYP1A2CYP3A4GAA
SCHEMBL5179725 0.78 ALDH1A1 (0.60) MAPTALDH1A1CYP1A2CYP3A4GAA
Hydrochloric Acid SCHEMBL2328872 0.77 SIRT2 (0.52) SIRT2SIRT1L3MBTL1CYP19A1CYP11B1
Hydrochloric Acid SCHEMBL2328868 0.77 SIRT2 (0.52) SIRT2SIRT1L3MBTL1CYP19A1CYP11B1
Hydrochloric Acid SCHEMBL5180312 0.77 ALDH1A1 (0.59) MAPTALDH1A1CYP1A2CYP3A4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853618-A4 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE POULENC RORER PHARMA (US) 2000-03-15 EP disclosed
EP-0853618-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1998-07-22 EP disclosed
US-5612353-A ANTICOAGULANT RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1997-03-18 US disclosed
WO-1996040679-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N-[(AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHÔNE-POULENC RORER PHARMACEUTICALS INC. (US) 1996-12-19 WO disclosed