SCHEMBL742022

SCHEMBL742022

COCCCn1c([C@@H]2CCCN(C(=O)[C@@H]3CN(C(=O)c4cccc(Cl)c4)C[C@H]3N)C2)nc2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 5/20 0.43
KCNH2 Q12809 3/20 0.43
HRH1 P35367 2/20 0.43
CYP2D6 P10635 1/20 0.43
PROKR1 Q8TCW9 4/20 0.43
CHRM1 P11229 1/20 0.43
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
DPP8 Q6V1X1 3/20 0.42
CNR2 P34972 1/20 0.41
HSD11B1 P28845 1/20 0.41
IRAK4 Q9NWZ3 1/20 0.41
ADORA2A P29274 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL742023 1.00 DPP4 (0.43) DPP4KCNH2HRH1CYP2D6PROKR1
SCHEMBL741961 0.92 HRH1 (0.45) DPP4KCNH2HRH1CYP2D6PROKR1
SCHEMBL741962 0.92 HRH1 (0.45) DPP4KCNH2HRH1CYP2D6PROKR1
SCHEMBL738833 0.92 HRH1 (0.49) DPP4KCNH2HRH1CYP2D6PROKR1
SCHEMBL738834 0.92 HRH1 (0.49) DPP4KCNH2HRH1CYP2D6PROKR1
SCHEMBL740546 0.92 DPP4 (0.44) DPP4KCNH2HRH1CYP2D6PROKR1
SCHEMBL740493 0.92 OPRK1 (0.43) DPP4KCNH2HRH1CYP2D6PROKR1
SCHEMBL740173 0.92 KCNH2 (0.47) DPP4KCNH2HRH1CYP2D6PROKR1
SCHEMBL740538 0.92 HRH1 (0.43) DPP4KCNH2HRH1CYP2D6PROKR1
SCHEMBL740174 0.92 KCNH2 (0.47) DPP4KCNH2HRH1CYP2D6PROKR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US claimed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed