SCHEMBL7422018

SCHEMBL7422018

COc1cc(CC(=O)NCC2CCN(C(=O)OC(C)(C)C)CC2)ccc1NC(=O)Nc1ccccc1C

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 3/20 0.51
KDM4E B2RXH2 1/20 0.50
PKM P14618 1/20 0.50
ITGA4 P13612 8/20 0.49
ITGB1 P05556 7/20 0.49
GPR119 Q8TDV5 2/20 0.46
BRD4 O60885 2/20 0.45
LMNA P02545 1/20 0.44
TP53 P04637 1/20 0.44
GNRHR P30968 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7427113 0.84 ITGA4 (0.47) ITGA4ITGB1
SCHEMBL7427128 0.84 ITGA4 (0.47) ITGA4ITGB1
SCHEMBL7425032 0.84 ITGA4 (0.64) ITGA4ITGB1LMNAL3MBTL1
SCHEMBL7389620 0.84 ITGA4 (0.53) ITGA4ITGB1
SCHEMBL7535332 0.83 ITGA4 (0.57) TGFBR1KDM4EITGA4ITGB1LMNA
SCHEMBL7394951 0.83 ITGA4 (0.54) ITGA4ITGB1BRD4L3MBTL1
SCHEMBL7430173 0.83 ITGA4 (0.54) ITGA4ITGB1
SCHEMBL7429572 0.82 ITGA4 (0.61) ITGA4ITGB1
SCHEMBL7426837 0.81 ITGA4 (0.60) KDM4EITGA4ITGB1L3MBTL1
SCHEMBL14558521 0.79 ITGA4 (0.57) ITGA4ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999054321-A1 SUBSTITUTED DIAMINES AND THEIR USE AS CELL ADHESION INHIBITORS AVENTIS PHARMA LIMITED (GB) 1999-10-28 WO disclosed