SCHEMBL7422939

SCHEMBL7422939

COC(=O)[C@@H](NC(=O)C=Cc1ccccc1)C(C)C

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.60
NOS2 P35228 8/20 0.57
NOS3 P29474 7/20 0.57
NOS1 P29475 7/20 0.57
ALDH1A1 P00352 2/20 0.54
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
MAPK1 P28482 1/20 0.53
CYP2C19 P33261 1/20 0.53
TAS1R3 Q7RTX0 2/20 0.52
TAS1R1 Q7RTX1 2/20 0.52
HDAC3 O15379 1/20 0.51
HDAC4 P56524 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
LMNA P02545 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7422933 1.00 TDP1 (0.60) TDP1NOS2NOS3NOS1ALDH1A1
SCHEMBL27391709 0.90 TDP1 (0.58) TDP1NOS2NOS3NOS1ALDH1A1
SCHEMBL27391707 0.90 TDP1 (0.58) TDP1NOS2NOS3NOS1ALDH1A1
SCHEMBL31389136 0.87 TDP1 (0.56) TDP1NOS2NOS3NOS1ALDH1A1
SCHEMBL10459919 0.87 NOS2 (0.48) TDP1NOS2NOS3NOS1ALDH1A1
SCHEMBL7425727 0.86 TDP1 (0.65) TDP1ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL7425739 0.86 TDP1 (0.65) TDP1ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL10807729 0.83 TDP1 (0.57) TDP1NOS2NOS3NOS1ALDH1A1
SCHEMBL10807719 0.83 TDP1 (0.57) TDP1NOS2NOS3NOS1ALDH1A1
SCHEMBL31414519 0.81 TTR (0.57) NOS2NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1152910-A Difluorostatone antiviral agents MERRELL PHARMA INC (US) 1997-06-25 CN disclosed
EP-0773926-A1 DIFLUOROSTATONE ANTIVIRAL AGENTS MERRELL PHARMACEUTICALS INC. (US) 1997-05-21 EP disclosed
WO-1996002499-A1 DIFLUOROSTATONE ANTIVIRAL AGENTS MERRELL PHARMACEUTICALS INC. (US) 1996-02-01 WO disclosed