SCHEMBL7423258

SCHEMBL7423258

O=C(O)c1ccc2c(c1)CCN(C(=O)C(F)(F)F)CC2

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.57
ESR2 Q92731 6/20 0.57
ALDH1A1 P00352 2/20 0.56
HDAC6 Q9UBN7 5/20 0.53
HDAC8 Q9BY41 1/20 0.46
MYC P01106 1/20 0.44
PKM P14618 1/20 0.41
ABHD6 Q9BV23 2/20 0.40
SRD5A2 P31213 2/20 0.40
SRD5A1 P18405 1/20 0.40
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
BLM P54132 1/20 0.39
GRM1 Q13255 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14101079 0.91 ESR1 (0.70) ESR1ESR2ALDH1A1HDAC6HDAC8
SCHEMBL1787035 0.87 ESR1 (0.56) ESR1ESR2HDAC6HDAC8PKM
SCHEMBL5418547 0.84 ESR1 (0.50) ESR1ESR2HDAC6HDAC8PKM
SCHEMBL1366408 0.83 ESR1 (0.52) ESR1ESR2ALDH1A1HDAC6HDAC8
SCHEMBL9052486 0.83 HDAC6 (0.59) ESR1ESR2ALDH1A1HDAC6HDAC8
SCHEMBL4075352 0.83 ESR1 (0.52) ESR1ESR2ALDH1A1HDAC6HDAC8
SCHEMBL12387505 0.83 ESR1 (0.52) ESR1ESR2HDAC6HDAC8PKM
SCHEMBL27812215 0.82 ALDH1A1 (0.65) ALDH1A1HDAC6HDAC8MYCSRD5A2
Hydrochloric Acid SCHEMBL2315162 0.82 ESR1 (0.51) ESR1ESR2HDAC6HDAC8PKM
SCHEMBL373697 0.81 ESR2 (0.83) ESR1ESR2HDAC6ABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777667-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT Dr. Karl Thomae GmbH (DE) 1997-06-11 EP disclosed
WO-1996005194-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT DR. KARL THOMAE GMBH (DE) 1996-02-22 WO disclosed