SCHEMBL7423474

SCHEMBL7423474

CC(C)CC(NCCC(C(=O)O)C(=O)Nc1nc2ccc(F)cc2s1)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.52
DYRK1A Q13627 1/20 0.52
ACP1 P24666 1/20 0.49
LRRK2 Q5S007 2/20 0.48
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 2/20 0.48
PTPN1 P18031 1/20 0.48
KMT2A Q03164 2/20 0.46
CSNK1D P48730 1/20 0.44
PAX8 Q06710 1/20 0.44
NPC1 O15118 6/20 0.44
RAB9A P51151 6/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
MAPT P10636 2/20 0.44
ALPL P05186 1/20 0.44
GAA P10253 1/20 0.44
HPGD P15428 1/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7421668 0.90 PDPK1 (0.54) PDPK1DYRK1AACP1LRRK2ALDH1A1
SCHEMBL5869988 0.80 PAX8 (0.54) PDPK1DYRK1AACP1LRRK2ALDH1A1
SCHEMBL5869979 0.80 PAX8 (0.54) PDPK1DYRK1AACP1LRRK2ALDH1A1
SCHEMBL5869910 0.80 PAX8 (0.54) PDPK1DYRK1AACP1LRRK2ALDH1A1
SCHEMBL5870315 0.79 PDPK1 (0.55) PDPK1DYRK1AACP1LRRK2ALDH1A1
SCHEMBL5870537 0.79 PDPK1 (0.55) PDPK1DYRK1AACP1LRRK2ALDH1A1
SCHEMBL7424266 0.79 DYRK1A (0.53) DYRK1AACP1ALDH1A1KDM4EPTPN1
SCHEMBL5870526 0.79 PDPK1 (0.55) PDPK1DYRK1AACP1LRRK2ALDH1A1
SCHEMBL7427256 0.78 DYRK1A (0.54) DYRK1AACP1ALDH1A1KDM4EPTPN1
SCHEMBL7421229 0.78 DYRK1A (0.54) DYRK1AACP1ALDH1A1KDM4EPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed