SCHEMBL7423841

SCHEMBL7423841

CCOC(=O)c1coc(CN2CCCC2)n1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.55
TSHR P16473 3/20 0.45
NPSR1 Q6W5P4 1/20 0.45
NLRP3 Q96P20 1/20 0.45
CACNA1G O43497 5/20 0.44
ELANE P08246 2/20 0.43
ALDH1A1 P00352 1/20 0.43
KDM4E B2RXH2 2/20 0.43
KCNH2 Q12809 2/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
CYP1A2 P05177 1/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
RXFP1 Q9HBX9 1/20 0.42
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3387830 0.99 HRH3 (0.57) HRH3TSHRNPSR1NLRP3CACNA1G
Maleic Acid SCHEMBL7427563 0.93 HRH3 (0.49) HRH3TSHRNPSR1NLRP3CACNA1G
Fumaric Acid SCHEMBL7427567 0.93 HRH3 (0.49) HRH3TSHRNPSR1NLRP3CACNA1G
SCHEMBL3384502 0.90 HRH3 (0.58) HRH3TSHRCACNA1GALDH1A1KDM4E
SCHEMBL7427115 0.86 HRH3 (0.57) HRH3NPSR1CACNA1GELANEALDH1A1
SCHEMBL7421852 0.85 HRH3 (0.59) HRH3NPSR1CACNA1GELANEALDH1A1
SCHEMBL7424821 0.80 HRH3 (0.59) HRH3CACNA1GELANEKCNH2RAB9A
Maleic Acid SCHEMBL7424004 0.80 CACNA1G (0.52) HRH3NPSR1CACNA1GELANEALDH1A1
Fumaric Acid SCHEMBL7424008 0.80 CACNA1G (0.52) HRH3NPSR1CACNA1GELANEALDH1A1
SCHEMBL9714181 0.79 CYP1A2 (0.51) TSHRNLRP3ALDH1A1KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000053589-A1 PROCESS FOR PREPARING OXAZOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 2000-09-14 WO disclosed
EP-1003748-A2 PYRROLOPYRROLONE DERIVATIVES AS INHIBITORS OF NEUTROPHIL ELASTASE GLAXO GROUP LIMITED (GB) 2000-05-31 EP disclosed
WO-1999012933-A2 PYRROLOPYRROLONE DERIVATIVES AS INHIBITORS OF NEUTROPHIL ELASTASE GLAXO GROUP LIMITED (GB) 1999-03-18 WO disclosed