SCHEMBL7424229

SCHEMBL7424229

[c]1cccc2c3c(ccc12)OCO3

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BAD Q92934 5/20 0.44
ABCG2 Q9UNQ0 1/20 0.35
ALDH1A1 P00352 4/20 0.35
CYP1A2 P05177 3/20 0.35
KDM4E B2RXH2 3/20 0.35
MAPT P10636 3/20 0.35
HPGD P15428 3/20 0.35
MAPK1 P28482 3/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
HSD17B10 Q99714 3/20 0.35
MEN1 O00255 2/20 0.35
LMNA P02545 2/20 0.35
KMT2A Q03164 2/20 0.35
RGS17 Q9UGC6 2/20 0.35
RGS12 O14924 2/20 0.35
TP53 P04637 2/20 0.35
BCHE P06276 2/20 0.35
CYP3A4 P08684 2/20 0.35
ALOX15 P16050 2/20 0.35
ALOX12 P18054 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7437286 0.76 ABCG2 (0.41) BADABCG2ALDH1A1CYP1A2KDM4E
SCHEMBL7426502 0.71 ABCG2 (0.35) BADABCG2ALDH1A1CYP1A2KDM4E
SCHEMBL2411016 0.71 CYP1A2 (0.32) CYP1A2
SCHEMBL7432722 0.70 ABCG2 (0.38) ABCG2ALDH1A1KDM4EMAPTHPGD
SCHEMBL30400843 0.69 BAD (0.49) BADABCG2ALDH1A1CYP1A2KDM4E
SCHEMBL403982 0.69 BAD (0.49) BADABCG2ALDH1A1CYP1A2KDM4E
SCHEMBL2412656 0.67 HPRT1 (0.33)
SCHEMBL2884931 0.66 ABCG2 (0.52) ABCG2SMN1; SMN2LMNACYP3A4PKM
SCHEMBL9871797 0.66 BAD (0.53) BADABCG2ALDH1A1CYP1A2KDM4E
SCHEMBL4894 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0283310-B1 N-BENZHYDRYL-SUBSTITUTED HETEROCYCLIC DERIVATIVES, THEIR PREPARATION AND THEIR USE Sankyo Company Limited (JP) 1993-05-26 EP disclosed
US-5028610-A Calcium Channel Blockers SANKYO COMPANY LIMITED (JP) 1991-07-02 US disclosed
EP-0283310-A1 N-Benzhydryl-substituted heterocyclic derivatives, their preparation and their use Sankyo Company Limited (JP) 1988-09-21 EP disclosed