SCHEMBL7424926

SCHEMBL7424926

CCOC(=O)/C=C(\N)CF

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.50
ALOX15 P16050 1/20 0.44
HCAR2 Q8TDS4 1/20 0.42
ALDH1A1 P00352 5/20 0.37
LMNA P02545 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MAPT P10636 2/20 0.35
GAA P10253 2/20 0.34
MGAM O43451 1/20 0.34
SI P14410 1/20 0.34
MGAM2 Q2M2H8 1/20 0.34
SOAT1 P35610 1/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
GLO1 Q04760 1/20 0.32
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7424929 1.00 NPSR1 (0.50) NPSR1ALOX15HCAR2ALDH1A1LMNA
SCHEMBL7913300 1.00 NPSR1 (0.50) NPSR1ALOX15HCAR2ALDH1A1LMNA
SCHEMBL7912959 0.83 NPSR1 (0.54) NPSR1ALOX15HCAR2ALDH1A1LMNA
SCHEMBL3190948 0.83 NPSR1 (0.54) NPSR1ALOX15HCAR2ALDH1A1LMNA
SCHEMBL4753860 0.83 NPSR1 (0.54) NPSR1ALOX15HCAR2ALDH1A1LMNA
SCHEMBL8201155 0.79 NPSR1 (0.50) NPSR1ALOX15HCAR2ALDH1A1LMNA
SCHEMBL1061977 0.79 NPSR1 (0.50) NPSR1ALOX15HCAR2ALDH1A1LMNA
SCHEMBL7598957 0.79 NPSR1 (0.46) NPSR1ALOX15HCAR2ALDH1A1LMNA
SCHEMBL24116900 0.78
SCHEMBL7428622 0.78

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4686217-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS FISONS PLC (GB) 1987-08-11 US disclosed
US-4607041-A CARDIOTONIC AGENTS FISONS PLC (GB) 1986-08-19 US disclosed
EP-0125803-A2 Pharmaceutically active dihydropyridines FISONS plc (GB) 1984-11-21 EP disclosed