SCHEMBL7424935

SCHEMBL7424935

Clc1ccc2[nH][c]cc2c1-c1ncc[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.39
MTOR P42345 1/20 0.39
ADK P55263 1/20 0.39
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP19A1 P11511 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
ADRA1A P35348 2/20 0.31
ADRA2A P08913 1/20 0.31
ADRA2C P18825 1/20 0.31
ADRA1D P25100 1/20 0.31
ADRA1B P35368 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6002606 0.71 ADRA2A (0.52) NISCHMTORADKALDH1A1KDM4E
SCHEMBL1719454 0.65 NISCH (0.53) NISCHMTORADKALDH1A1KDM4E
SCHEMBL5886380 0.65 NISCH (0.39) NISCHMTORADKALDH1A1KDM4E
SCHEMBL24575956 0.64 CCR1 (0.42) NISCHMTORADKALDH1A1KDM4E
SCHEMBL206251 0.64 HRH4 (0.33)
SCHEMBL1288554 0.62 NISCH (0.52) NISCHMTORADKALDH1A1KDM4E
SCHEMBL482165 0.62 NISCH (0.64) NISCHMTORADKALDH1A1KDM4E
SCHEMBL722191 0.61 NISCH (0.78) NISCHMTORADKALDH1A1KDM4E
SCHEMBL14663248 0.61 NISCH (0.39) NISCHMTORADKALDH1A1KDM4E
SCHEMBL8540910 0.61 NISCH (0.50) NISCHMTORADKALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1082321-A1 HETEROCYCLIC DERIVATIVES WHICH INHIBIT FACTOR XA AstraZeneca AB (SE) 2001-03-14 EP disclosed
WO-1999057113-A1 HETEROCYCLIC DERIVATIVES WHICH INHIBIT FACTOR XA ASTRAZENECA AB (SE) 1999-11-11 WO disclosed