SCHEMBL7425232

SCHEMBL7425232

Cc1ccc(C#N)c(F)c1Br

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.40
TRPV4 Q9HBA0 1/20 0.35
AR P10275 6/20 0.34
EGLN2 Q96KS0 3/20 0.33
CYP11B1 P15538 3/20 0.33
CYP11B2 P19099 3/20 0.33
ALDH1A1 P00352 1/20 0.33
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
NOTUM Q6P988 1/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3882893 0.80 TSHR (0.44) TSHRARALDH1A1MAOAMAOB
SCHEMBL410450 0.80 TSHR (0.44) TSHRTRPV4AREGLN2CYP11B1
SCHEMBL13199476 0.78 TSHR (0.43) TSHRTRPV4AREGLN2CYP11B1
SCHEMBL17545789 0.77 TSHR (0.41) TSHRTRPV4AREGLN2CYP11B1
SCHEMBL19628965 0.75 AR (0.41) TSHRTRPV4ARALDH1A1
SCHEMBL152425 0.75 AR (0.40) TSHRTRPV4AREGLN2CYP11B1
SCHEMBL21860014 0.75 AR (0.41) TSHRTRPV4ARALDH1A1
SCHEMBL1222533 0.75 TSHR (0.40) TSHRTRPV4AREGLN2CYP11B1
SCHEMBL28201225 0.75 TSHR (0.40) TSHRTRPV4AREGLN2CYP11B1
SCHEMBL26094546 0.75 TSHR (0.40) TSHRARALDH1A1MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024099269-A1 ARYLAMIDE COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, USE THEREOF 华东师范大学 2024-05-16 WO disclosed
CN-118026880-A Aryl amide compound, pharmaceutical composition containing same and application thereof 华东师范大学 2024-05-14 CN disclosed
WO-2001079195-A2 PYRIDINE AND PYRAZINE DERIVATIVES AS THROMBIN INHIBITORS CORVAS INTERNATIONAL, INC. (US) 2001-10-25 WO disclosed
WO-2001079193-A2 SUBSTITUTED HYDRAZINYL HETEROAROMATIC INHIBITORS OF THROMBIN CORVAS INTERNATIONAL, INC. (US) 2001-10-25 WO disclosed
WO-2001079261-A1 TETRAHYDRO-AZEPINONE DERIVATIVES AS THROMBIN INHIBITORS CORVAS INTERNATIONAL, INC. (US) 2001-10-25 WO disclosed