SCHEMBL7425451

SCHEMBL7425451

N[C@@H](Cc1nc2ccccc2s1)C(=O)N1CCN(CCF)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.47
DRD3 P35462 6/20 0.47
DRD4 P21917 5/20 0.47
HTR7 P34969 6/20 0.44
HTR1A P08908 5/20 0.44
HRH1 P35367 3/20 0.44
ADRA2A P08913 2/20 0.44
ADRA2C P18825 2/20 0.44
SLC6A2 P23975 2/20 0.44
ADRA1A P35348 2/20 0.44
HTR2B P41595 2/20 0.44
SIGMAR1 Q99720 1/20 0.44
HTR2A P28223 5/20 0.43
F2 P00734 1/20 0.43
POLB P06746 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MAPT P10636 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
PKM P14618 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL7425687 0.99 DRD2 (0.46) DRD2DRD3DRD4HTR7HTR1A
Bromide SCHEMBL7418489 0.99 DRD2 (0.46) DRD2DRD3DRD4HTR7HTR1A
Bromide SCHEMBL7418493 0.99 DRD2 (0.46) DRD2DRD3DRD4HTR7HTR1A
Bromide SCHEMBL7425690 0.99 DRD2 (0.46) DRD2DRD3DRD4HTR7HTR1A
SCHEMBL7419443 0.94 DRD2 (0.50) DRD2DRD3DRD4HTR7HTR1A
SCHEMBL7426173 0.87 PRMT5 (0.44) DRD2DRD3DRD4HTR7HTR1A
Hydrochloric Acid SCHEMBL7422561 0.86 NPC1 (0.52) DRD2DRD3DRD4F2POLB
SCHEMBL7426600 0.85 DRD2 (0.46) DRD2DRD3DRD4HTR7HTR1A
SCHEMBL7360493 0.84 F2 (0.53) F2
SCHEMBL7359256 0.84 F2 (0.53) F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0815103-A1 TRYPSIN AND THROMBIN INHIBITORS Novartis AG (CH) 1998-01-07 EP disclosed
WO-1997046553-A1 THROMBIN INHIBITORS NOVARTIS AG (CH) 1997-12-11 WO disclosed
WO-1996029327-A1 TRYPSIN AND THROMBIN INHIBITORS NOVARTIS AG (CH) 1996-09-26 WO disclosed