SCHEMBL7425945

SCHEMBL7425945

O=S(=O)(O)c1ccc(-c2cccnc2)s1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 2/20 0.55
MKNK2 Q9HBH9 2/20 0.55
CYP2A6 P11509 13/20 0.54
CYP2C19 P33261 8/20 0.54
CYP2C9 P11712 8/20 0.54
CYP3A4 P08684 7/20 0.54
CYP2E1 P05181 6/20 0.53
CYP2B6 P20813 6/20 0.53
CYP2D6 P10635 6/20 0.53
HDAC3 O15379 1/20 0.53
HDAC4 P56524 1/20 0.53
HDAC1 Q13547 1/20 0.53
HDAC7 Q8WUI4 1/20 0.53
HDAC2 Q92769 1/20 0.53
HDAC10 Q969S8 1/20 0.53
HDAC11 Q96DB2 1/20 0.53
HDAC8 Q9BY41 1/20 0.53
HDAC6 Q9UBN7 1/20 0.53
HDAC9 Q9UKV0 1/20 0.53
HDAC5 Q9UQL6 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27502977 0.98 MKNK1 (0.54) MKNK1MKNK2CYP2A6CYP2C19CYP2C9
SCHEMBL364159 0.83 CYP2A6 (0.57) MKNK1MKNK2CYP2A6CYP2C19CYP2C9
SCHEMBL7425364 0.81 HDAC3 (0.49) CYP2C19CYP2C9CYP3A4CYP2D6HDAC3
SCHEMBL3046411 0.80 RAB9A (0.47) CYP2A6CYP2C19CYP2C9CYP3A4CYP2E1
Pyridine SCHEMBL28017964 0.80 CYP2A6 (0.53) MKNK1MKNK2CYP2A6CYP2C19CYP2C9
Hydrochloric Acid SCHEMBL27503318 0.79 HDAC3 (0.47) CYP2C19CYP2C9CYP3A4CYP2D6HDAC3
SCHEMBL29854440 0.78 CYP2A6 (0.73) MKNK1MKNK2CYP2A6CYP2C19CYP2C9
SCHEMBL7423572 0.76 MKNK1 (0.41) MKNK1MKNK2CYP2A6CNR1
SCHEMBL7054825 0.76 RAB9A (0.51) HDAC1HDAC6ALDH1A1CYP1A2CA12
SCHEMBL7213572 0.74 DYRK1A (0.58) MKNK1MKNK2CYP2A6CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1244798-A Sulfonic acid or sulfonylamino N-(heteroaralkyl)-azaheterocyclylamide compounds RHONE POULENC RORER PHARMA (US) 2000-02-16 CN claimed
CN-1418882-A Substituted sulfonic acid N- [ (aminoiminomethyl) phenylalkyl ] -azacyclic amide compounds AVENTIS PHARMACENEITCALS INC (US) 2003-05-21 CN disclosed
CN-1093856-C Substituted sulfonic acid N- [ (aminoiminomethyl) phenylalkyl ] -azacyclic amide compounds AVENTIS PHARM PROD INC (US) 2002-11-06 CN disclosed
EP-0894088-A4 SUBSTITUTED SULFONIC ACID N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLAMIDE COMPOUNDS RHONE POULENC RORER PHARMA (US) 2001-12-05 EP disclosed
US-6034093-A Substituted sulfonic acid N-[(aminoiminomethyl)phenylalkyl]-azaheterocyclylamide compounds RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 2000-03-07 US disclosed
CN-1244798-A Sulfonic acid or sulfonylamino N-(heteroaralkyl)-azaheterocyclylamide compounds RHONE POULENC RORER PHARMA (US) 2000-02-16 CN disclosed
CN-1213370-A Substituted sulfonic acid N- [ (aminoiminomethyl) phenylalkyl ] -azacyclic amide compounds RHONE POULENC RORER PHAMACEUTI (US) 1999-04-07 CN disclosed
EP-0894088-A1 SUBSTITUTED SULFONIC ACID N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLAMIDE COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1999-02-03 EP disclosed
WO-1998024784-A1 SUBSTITUTED SULFONIC ACID N-[(AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLAMIDE COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-06-11 WO disclosed
US-5731315-A Substituted sulfonic acid n- (aminoiminomethyl)phenylalkyl!-azaheterocyclamide compounds RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-03-24 US disclosed