SCHEMBL7428693

SCHEMBL7428693

C[C@@H]1Cc2cc(Br)ccc2NC1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.51
ADRA2A P08913 3/20 0.42
PNMT P11086 3/20 0.42
ADRA2B P18089 3/20 0.42
ADRA2C P18825 3/20 0.42
GABRA1 P14867 1/20 0.42
GABRA5 P31644 1/20 0.42
GABRA3 P34903 1/20 0.42
GABRA2 P47869 1/20 0.42
GABRB2 P47870 1/20 0.42
CMA1 P23946 1/20 0.41
AHR P35869 1/20 0.41
TDP2 O95551 1/20 0.39
TP53 P04637 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
TGM2 P21980 1/20 0.39
CES1 P23141 1/20 0.39
LMNA P02545 1/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14550603 1.00 BRD4 (0.51) BRD4ADRA2APNMTADRA2BADRA2C
SCHEMBL1347544 0.84 BRD4 (0.49) BRD4ADRA2APNMTADRA2BADRA2C
SCHEMBL434007 0.81 ACHE (0.49) BRD4POLBPKMPDE3BPDE3A
SCHEMBL18743294 0.81 ACHE (0.49) BRD4POLBPKMPDE3BPDE3A
SCHEMBL14721601 0.80 CA9 (0.40) BRD4MAPTLMNAPDE3BPDE3A
SCHEMBL4596331 0.80 BRD4 (0.47) BRD4ADRA2APNMTADRA2BADRA2C
SCHEMBL7866698 0.80 AHR (0.53) ADRA2AADRA2BADRA2CCMA1AHR
SCHEMBL5131215 0.80 BRD4 (0.47) BRD4ADRA2APNMTADRA2BADRA2C
SCHEMBL31398247 0.80 BRD4 (0.44) BRD4ADRA2APNMTADRA2BADRA2C
Hydrochloric Acid SCHEMBL25330756 0.79 BRD4 (0.46) BRD4ADRA2APNMTADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0815103-A1 TRYPSIN AND THROMBIN INHIBITORS Novartis AG (CH) 1998-01-07 EP disclosed
WO-1996029327-A1 TRYPSIN AND THROMBIN INHIBITORS NOVARTIS AG (CH) 1996-09-26 WO disclosed