SCHEMBL7429785

SCHEMBL7429785

CC(C)c1nc(CNC(=O)N[C@H](C(=O)O)C(C)C)cs1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.50
TSHR P16473 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.43
HSD17B10 Q99714 1/20 0.42
ADORA2A P29274 1/20 0.42
ALDH1A1 P00352 4/20 0.41
CYP3A4 P08684 3/20 0.40
SLC6A3 Q01959 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7424264 0.87 MEN1 (0.52) SMN1; SMN2HSD17B10ADORA2AALDH1A1CYP3A4
SCHEMBL7395069 0.81 ALDH1A1 (0.42) ALDH1A1CYP3A4SLC6A3MEN1KMT2A
SCHEMBL27900691 0.80 CYP3A4 (0.56) CYP3A4
SCHEMBL1389204 0.80 CYP3A4 (0.56) CYP3A4
SCHEMBL7178746 0.80 CYP3A4 (0.48) CYP3A4
SCHEMBL7391613 0.80 CYP3A4 (0.56) CYP3A4
SCHEMBL7178744 0.80 CYP3A4 (0.48) CYP3A4
SCHEMBL7527628 0.79 CYP3A4 (0.55) CYP3A4
SCHEMBL7188807 0.78 CYP3A4 (0.44) CYP3A4
SCHEMBL7178210 0.78 CYP3A4 (0.43) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008103949-A1 MODULATORS OF PHARMACOKINETIC PROPERTIES OF THERAPEUTICS GILEAD SCIENCES, INC. (US) 2008-08-28 WO disclosed
EP-1077977-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 2001-02-28 EP disclosed
WO-1999059994-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1999-11-25 WO disclosed