SCHEMBL7430359

SCHEMBL7430359

Fc1cccnc1-c1cccs1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.47
CYP11B2 P19099 1/20 0.47
CYP2C9 P11712 2/20 0.44
CYP2E1 P05181 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2A6 P11509 1/20 0.44
CYP2B6 P20813 1/20 0.44
TDO2 P48775 1/20 0.43
CDK5 Q00535 1/20 0.43
CDK5R1 Q15078 1/20 0.43
PDE3B Q13370 1/20 0.43
PDE3A Q14432 1/20 0.43
RPS6KB2 Q9UBS0 3/20 0.42
CYP19A1 P11511 1/20 0.41
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 3/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HPGD P15428 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4170768 0.78 CYP11B1 (0.48) CYP11B1CYP11B2CYP2C9CYP2E1CYP3A4
SCHEMBL29675365 0.78 CYP11B1 (0.48) CYP11B1CYP11B2CYP2C9CYP2E1CYP3A4
SCHEMBL30497068 0.77 CYP11B1 (0.47) CYP11B1CYP11B2CYP2C9CYP2E1CYP3A4
SCHEMBL28931076 0.77 CYP11B1 (0.47) CYP11B1CYP11B2CYP2C9CYP2E1CYP3A4
SCHEMBL28549409 0.77 CYP11B1 (0.47) CYP11B1CYP11B2CYP2C9CYP2E1CYP3A4
SCHEMBL10670524 0.77 CYP11B1 (0.50) CYP11B1CYP11B2CYP2C9CYP2E1CYP3A4
SCHEMBL4974064 0.77 RPS6KB2 (0.53) CYP11B1CYP11B2CYP2C9CYP2E1CYP3A4
SCHEMBL3831303 0.77 TRPV1 (0.44) CYP11B1CYP11B2CYP2C9CYP2E1CYP3A4
SCHEMBL15624391 0.76 TDP1 (0.44) CYP3A4KDM4EMAPTMEN1KMT2A
SCHEMBL2455860 0.76 CYP11B1 (0.46) CYP11B1CYP11B2CYP2C9CYP2E1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002000623-A2 ARYL FUSED SUBSTITUTED 4-OXY-PYRIDINES NEUROGEN CORPORATION (US) 2002-01-03 WO claimed
WO-2002000623-A2 ARYL FUSED SUBSTITUTED 4-OXY-PYRIDINES NEUROGEN CORPORATION (US) 2002-01-03 WO disclosed