SCHEMBL2455860

SCHEMBL2455860

c1csc(-c2ncccc2[Ir]c2cccnc2-c2cccs2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
CYP2E1 P05181 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2A6 P11509 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2B6 P20813 1/20 0.43
CDK5 Q00535 2/20 0.42
CDK5R1 Q15078 2/20 0.42
TDO2 P48775 1/20 0.42
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
RPS6KB2 Q9UBS0 3/20 0.41
CYP19A1 P11511 1/20 0.40
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29675365 0.77 CYP11B1 (0.48) CYP11B1CYP11B2CYP2E1CYP3A4CYP2A6
SCHEMBL4170768 0.77 CYP11B1 (0.48) CYP11B1CYP11B2CYP2E1CYP3A4CYP2A6
SCHEMBL28549409 0.76 CYP11B1 (0.47) CYP11B1CYP11B2CYP2E1CYP3A4CYP2A6
SCHEMBL10670524 0.76 CYP11B1 (0.50) CYP11B1CYP11B2CYP2E1CYP3A4CYP2A6
SCHEMBL4974064 0.76 RPS6KB2 (0.53) CYP11B1CYP11B2CYP2E1CYP3A4CYP2A6
SCHEMBL30497068 0.76 CYP11B1 (0.47) CYP11B1CYP11B2CYP2E1CYP3A4CYP2A6
SCHEMBL28931076 0.76 CYP11B1 (0.47) CYP11B1CYP11B2CYP2E1CYP3A4CYP2A6
SCHEMBL7430359 0.76 CYP11B1 (0.47) CYP11B1CYP11B2CYP2E1CYP3A4CYP2A6
SCHEMBL2461437 0.74 CYP11B1 (0.46) CYP11B1CYP11B2CYP2E1CYP3A4CYP2A6
SCHEMBL3831303 0.71 TRPV1 (0.44) CYP11B1CYP11B2CYP2E1CYP3A4CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122094955-A Compound, light-emitting device, display device, electronic apparatus, and lighting device 2026-05-26 CN disclosed
US-20260059938-A1 ORGANIC EL ELEMENT, DISPLAY DEVICE, AND ILLUMINATION DEVICE TORAY INDUSTRIES, INC. (JP) 2026-02-26 US disclosed
EP-4656637-A1 COMPOUND, AND LIGHT-EMITTING ELEMENT, DISPLAY DEVICE, LIGHTING DEVICE AND PHOTOSENSITIZER EACH CONTAINING SAME Toray Industries, Inc. (JP) 2025-12-03 EP disclosed
WO-2025110081-A1 COMPOUND, LIGHT-EMITTING ELEMENT CONTAINING SAME, DISPLAY DEVICE, AND ILLUMINATION DEVICE 東レ株式会社 2025-05-30 WO disclosed
EP-4559914-A1 COMPOUND, LIGHT-EMITTING ELEMENT, DISPLAY DEVICE, AND LIGHTING DEVICE Toray Industries, Inc. (JP) 2025-05-28 EP disclosed
US-20250169275-A1 ORGANIC EL ELEMENT MATERIAL, ORGANIC EL ELEMENT, DISPLAY DEVICE AND ILLUMINATION DEVICE TORAY INDUSTRIES, INC. (JP) 2025-05-22 US disclosed
CN-114746402-B Compound, organic thin film light-emitting element, display device, and lighting device 东丽株式会社 2025-04-08 CN disclosed
WO-2025053127-A1 COMPOUND, ORGANIC ELECTROLUMINESCENT ELEMENT, DISPLAY DEVICE, AND LIGHTING DEVICE 東レ株式会社 2025-03-13 WO disclosed
CN-119546606-A Compound, light-emitting element, display device, and lighting device 东丽株式会社 2025-02-28 CN disclosed
WO-2025033193-A1 COMPOUND, LIGHT-EMITTING ELEMENT CONTAINING SAME, DISPLAY DEVICE, AND ILLUMINATION DEVICE 東レ株式会社 2025-02-13 WO disclosed
US-20150084020-A1 LIGHT-EMITTING DEVICE MATERIAL AND LIGHT-EMITTING DEVICE TORAY INDUSTRIES, INC. (JP) 2015-03-26 US disclosed
US-20140070204-A1 LIGHT EMITTING DEVICE MATERIAL AND LIGHT EMITTING DEVICE TORAY INDUSTRIES, INC. (JP) 2014-03-13 US disclosed
US-20130264558-A1 LIGHT EMITTING DEVICE MATERIAL AND LIGHT EMITTING DEVICE TORAY INDUSTRIES, INC. (JP) 2013-10-10 US disclosed
EP-2365735-B1 Luminescent element material and luminescent element comprising the same TORAY INDUSTRIES (JP) 2013-08-28 EP disclosed
EP-2365735-A2 Luminescent element material and luminescent element comprising the same TORAY INDUSTRIES INC. (JP) 2011-09-14 EP disclosed
US-7318966-B2 Luminescent element material and luminescent element comprising the same TORAY INDUSTRIES, INC. (JP) 2008-01-15 US disclosed
US-20060051615-A1 Organic electroluminescent element SANYO ELECTRIC CO., LTD. (JP) 2006-03-09 US disclosed
US-20060029828-A1 Organic electroluminescent device SANYO ELECTRIC CO., LTD. (JP) 2006-02-09 US disclosed
US-20030168970-A1 Luminescent element material and luminescent element comprising the same TORAY INDUSTRIES, INC. (JP) 2003-09-11 US disclosed
EP-1341403-A1 LUMINESCENT ELEMENT MATERIAL AND LUMINESCENT ELEMENT COMPRISING THE SAME Toray Industries, Inc. (JP) 2003-09-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030168970-A1 Luminescent element material and luminescent element comprising the same SAAL1, EBPL, CSNK1A1L CYP11B1 4309/4885CYP11B2 3963/4885CYP2E1 1991/4885
US-20260059938-A1 ORGANIC EL ELEMENT, DISPLAY DEVICE, AND ILLUMINATION DEVICE LEF1, LAGE3, EMC1 CYP11B1 1367/4885CYP11B2 1130/4885CYP2E1 1757/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.