SCHEMBL743053

SCHEMBL743053

O=C(O)N1CC2CN(Cc3c[nH]c4cc(Oc5nc6ccccc6s5)ccc34)CC2C1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 18/20 0.51
EPHX2 P34913 1/20 0.51
KCNH2 Q12809 4/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
SOS1 Q07889 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL744898 0.93 LTA4H (0.52) LTA4HEPHX2KCNH2
SCHEMBL742274 0.90 LTA4H (0.48) LTA4HEPHX2KCNH2
SCHEMBL745544 0.87 LTA4H (0.51) LTA4HEPHX2KCNH2
Hydrochloric Acid SCHEMBL3746254 0.86 LTA4H (0.50) LTA4HEPHX2KCNH2
SCHEMBL15252243 0.85 LTA4H (0.47) LTA4HEPHX2KCNH2
SCHEMBL743395 0.84 LTA4H (0.71) LTA4HEPHX2KCNH2
SCHEMBL744389 0.84 LTA4H (0.59) LTA4HEPHX2KCNH2
SCHEMBL15252290 0.83 LTA4H (0.59) LTA4HEPHX2KCNH2
SCHEMBL743354 0.83 LTA4H (0.59) LTA4HEPHX2KCNH2
SCHEMBL15252064 0.83 LTA4H (0.53) LTA4HEPHX2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430019-A1 COMPOUNDS WITH TWO FUSED BICYCLIC HETEROARYL MOIETIES AS MODULATORS OF LEUKOTRIENE A4 HYDROLASE Janssen Pharmaceutica, N.V. (BE) 2012-03-21 EP disclosed
WO-2010132599-A1 COMPOUNDS WITH TWO FUSED BICYCLIC HETEROARYL MOIETIES AS MODULATORS OF LEUKOTRIENE A4 HYDROLASE JANSSEN PHARMACEUTICA NV (BE) 2010-11-18 WO disclosed