SCHEMBL7432000

SCHEMBL7432000

CN1C(=O)C(N(C(=O)O)c2ccc([N+](=O)[O-])cc2)N=C(c2ccccc2)c2ccccc21

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 15/20 0.61
CCKAR P32238 3/20 0.52
GABRP O00591 1/20 0.49
GABRD O14764 1/20 0.49
GABRA1 P14867 1/20 0.49
GABRB1 P18505 1/20 0.49
GABRG2 P18507 1/20 0.49
GABRB3 P28472 1/20 0.49
GABRA5 P31644 1/20 0.49
GABRA3 P34903 1/20 0.49
GABRA2 P47869 1/20 0.49
GABRB2 P47870 1/20 0.49
GABRA4 P48169 1/20 0.49
GABRE P78334 1/20 0.49
GABRA6 Q16445 1/20 0.49
GABRG1 Q8N1C3 1/20 0.49
GABRG3 Q99928 1/20 0.49
GABRQ Q9UN88 1/20 0.49
LMNA P02545 1/20 0.45
OPRK1 P41145 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9718390 1.00 CCKBR (0.61) CCKBRCCKARGABRPGABRDGABRA1
SCHEMBL3252895 0.83 KCNH2 (0.47) CCKBR
SCHEMBL9867739 0.82 CCKBR (0.58) CCKBRCCKARGABRPGABRDGABRA1
SCHEMBL10683374 0.79 CCKBR (0.56) CCKBRCCKARGABRPGABRDGABRA1
SCHEMBL10520112 0.78 CCKBR (0.59) CCKBRCCKARGABRPGABRDGABRA1
Hydrochloric Acid SCHEMBL8926212 0.77 CCKBR (0.52) CCKBRCCKARGABRPGABRDGABRA1
Hydrochloric Acid SCHEMBL7206771 0.77 CCKBR (0.52) CCKBRCCKARGABRPGABRDGABRA1
SCHEMBL9866438 0.76 CCKBR (1.00) CCKBR
SCHEMBL9423126 0.74 CCKBR (0.74) CCKBRCCKAR
SCHEMBL9422961 0.74 CCKBR (0.74) CCKBRCCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175159-A Prevention of premature labor MERCK & CO., INC. (US) 1992-12-29 US disclosed
EP-0421802-A2 3-substituted-1,4-benzodiazepines useful as oxytocin antagonists MERCK & CO. INC. (US) 1991-04-10 EP disclosed