SCHEMBL7433158

SCHEMBL7433158

CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(O)=S

nearest known ligand 0.67

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSS P25774 9/20 0.67
CTSK P43235 8/20 0.67
CTSB P07858 2/20 0.67
CTSL P07711 1/20 0.67
ACE P12821 1/20 0.64
ATM Q13315 1/20 0.59
AKT1 P31749 1/20 0.58
KLK5 Q9Y337 1/20 0.56
PPARA Q07869 2/20 0.55
PPARG P37231 1/20 0.55
APP P05067 1/20 0.54
REN P00797 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6578977 1.00 CTSS (0.67) CTSSCTSKCTSBCTSLACE
SCHEMBL7271824 0.95 PPARA (0.63) CTSSCTSKCTSBCTSLACE
SCHEMBL2174152 0.89 CTSS (0.64) CTSSCTSKCTSBCTSLACE
SCHEMBL6473855 0.89 CTSS (0.64) CTSSCTSKCTSBCTSLACE
SCHEMBL795685 0.88 ACE (0.79) CTSSCTSKCTSBCTSLACE
SCHEMBL21473784 0.88 ACE (0.79) CTSSCTSKCTSBCTSLACE
SCHEMBL606309 0.88 ACE (0.79) CTSSCTSKCTSBCTSLACE
SCHEMBL7269746 0.88 CTSS (0.70) CTSSCTSKCTSBCTSLACE
SCHEMBL66220 0.88 ACE (0.79) CTSSCTSKCTSBCTSLACE
SCHEMBL67020 0.88 ACE (0.79) CTSSCTSKCTSBCTSLACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0604184-B1 Inhibitors of HIV protease useful for the treatment of aids LILLY CO ELI (US) 1997-07-09 EP disclosed
US-5554653-A Inhibitors of HIV protease useful for the treatment of AIDS ELI LILLY AND COMPANY (US) 1996-09-10 US disclosed
EP-0604184-A1 Inhibitors of HIV protease useful for the treatment of aids ELI LILLY AND COMPANY (US) 1994-06-29 EP disclosed
EP-0038117-A1 Methods for preparing anti-hypertensive agents UNIVERSITY OF MIAMI (US) 1981-10-21 EP disclosed