SCHEMBL7433456

SCHEMBL7433456

N=C(N)c1ccc(Cn2c(=O)ccc3cc(Oc4cccc(C(=N)N)c4)ccc32)cc1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
F10 P00742 12/20 0.56
F2 P00734 10/20 0.56
PRSS1 P07477 2/20 0.56
FURIN P09958 1/20 0.47
PLG P00747 2/20 0.46
PLAU P00749 2/20 0.46
ST14 Q9Y5Y6 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7420549 0.93 F2 (0.60) F10F2PRSS1FURINST14
SCHEMBL7430809 0.87 F2 (0.63) F10F2
SCHEMBL7433462 0.82 F10 (0.48) F10F2PRSS1FURIN
SCHEMBL7423194 0.81 F2 (0.67) F10F2
SCHEMBL7429823 0.80 F10 (0.60) F10F2PRSS1PLGPLAU
SCHEMBL7423757 0.79 F2 (0.61) F10F2PRSS1
SCHEMBL7432559 0.79 F10 (0.54) F10F2PLGPLAU
SCHEMBL7430906 0.79 F10 (0.67) F10F2PRSS1
SCHEMBL7426338 0.78 F10 (0.61) F10F2PRSS1PLAU
SCHEMBL7425222 0.78 F10 (0.47) F10F2PRSS1FURIN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1107954-A1 2-OXO-$i(2H)-QUINOLINE DERIVATIVES MERCK PATENT GmbH (DE) 2001-06-20 EP disclosed
WO-2000012479-A1 2-OXO-2H-QUINOLINE DERIVATIVES MERCK PATENT GMBH (DE) 2000-03-09 WO disclosed